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3-methyl-8-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-chloro-N,N-dimethyl-3-{[3-(propan-2-yl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpiperidin-4-amine
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,N-diethylpyrrolidin-3-amine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-chlorophenyl)propan-1-one
3-(3-methylphenyl)-1-(4-methylphenyl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
1-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-yl)benzamide
3-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-1-[3-(4-methylphenyl)phenyl]urea
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{[2-amino-6-(2-fluoro-5-methoxyphenyl)pyrimidin-4-yl]amino}ethan-1-ol
7-methyl-2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
6-(2-hydroxyethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-(furan-2-yl)-2-[4-(4-phenylpiperazine-1-carbonyl)-5-(propan-2-yl)-1H-pyrazol-1-yl]pyrimidine
3-acetyl-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
N,N-dimethyl-2-({[(1R,2R)-2-phenylcyclopropyl]formamido}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-ethyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-methyl-1H-pyrazole-5-carboxamide
2-[4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)morpholin-3-yl]-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
2,4-dimethyl-N-[4-(4-{[(4-phenyloxan-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
methyl 7-oxo-9-[2-(thiophen-3-yl)ethoxy]-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
7-(3-methoxypyridine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1,3-dimethyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
4-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]benzonitrile
2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]pyridine-4-carboxylic acid
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
methyl 1-[(1-ethylpyrrolidin-2-yl)methyl]-2-oxo-3-(pyridin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
ethyl 1-(3-acetamidopropanoyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(4aS,8aR)-6-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-cyclopropyl-N-[2-(3,4-dimethylphenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
6-chloro-2-[3-(pyridin-2-yl)azetidin-1-yl]-1,3-benzothiazole
1-methyl-4-(4-methyl-1H-imidazole-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[4-(5-chlorothiophene-2-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-(5-chloro-2-methoxyphenyl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-3-yl]propanamide
N-[(3S,4R)-1-(1H-indazole-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
3-{[1-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-N-[2-(dimethylamino)ethyl]benzamide
1-{4-[4-(2,3-dihydro-1H-isoindole-2-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
2-methoxy-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonitrile
2-{5-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
N-{[4-(methylsulfanyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
1-benzyl-4-{[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-cyclohexylpiperidine-4-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-3-phenylpropanamide
5,6-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}[(4-fluorophenyl)methyl]amine
4-[2-(carboxymethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzoic acid
4-{4-[2-fluoro-6-(propan-2-yloxy)phenyl]phenyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine