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N-(2-fluoro-5-methylphenyl)-4-(2-methyl-5-oxo-1,4-diazepan-1-yl)-4-oxobutanamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-{4-[(4-ethoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
1-methyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-(1H-imidazol-2-ylmethyl)cyclopropanamine
(4aR,7aS)-1-(2-ethylbutanoyl)-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3S,4R)-4-(4-methylphenyl)-1-[2-(2-methylphenyl)acetyl]pyrrolidin-3-yl]acetamide
6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
(3R,4S)-1-[(3-methylphenyl)methanesulfonyl]-4-(propan-2-yl)pyrrolidin-3-amine
8-({[(2-methylphenyl)methyl]carbamoyl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-methyl-1H-pyrrole-3-carboxamide
[1-(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-yl]methanol
N'-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pentanediamide
4-acetyl-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}benzene-1-sulfonamide
6-(2,5-dimethylfuran-3-yl)-8-oxo-7-(prop-2-en-1-yl)-N-(1,3-thiazol-2-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[2-(pyridin-4-yl)ethyl]-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
(3aR,6aR)-2-(5-ethylthiophene-2-carbonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
3-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[(3R,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
N-methyl-3-(2-oxo-1,2-dihydropyridin-1-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
(1R,2S)-1-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}-2,3-dihydro-1H-inden-2-ol
N-(2-methylpropyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-(piperidin-1-yl)-N1-(quinolin-6-yl)piperidine-1,4-dicarboxamide
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-(1-{[1-(pyrimidin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5-{[(2,6-dimethylpyridin-4-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-chloro-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-2-carboxamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(1-methyl-1H-pyrrol-2-yl)-2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethane-1,2-dione
1-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-(1H-imidazol-2-ylmethyl)-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 3-[2-oxo-6-(pyridin-4-ylmethoxy)-4-[3-(trifluoromethyl)benzoyl]-1,4-diazepan-1-yl]propanoate
N,N-dimethyl-7-(2,3,4-trimethoxybenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(5,6-dimethylpyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-[3-(pyridin-3-yl)azetidine-1-carbonyl]piperidine-1-carboxamide
3-hydroxy-N-(1-methyl-1H-pyrazol-4-yl)-3-(2-methylphenyl)pyrrolidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-(piperidin-1-ylmethyl)benzamide
2-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-1,4-dihydroquinolin-4-one
(3R)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
5-benzoyl-N-cyclopentyl-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{2-[1-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(2E)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-(quinolin-2-ylmethyl)prop-2-enamide
3-(5-{1H-pyrrolo[2,3-b]pyridine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
5-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-N-methylpyrimidin-2-amine