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3-[2-(dimethylamino)ethyl]-8-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)urea
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
3-({2-[1-(propan-2-yl)piperidin-4-yl]acetamido}methyl)-1,2,4-oxadiazole-5-carboxamide
(3S,9aR)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-methanesulfonyl-4-(piperidin-3-yl)-2-(pyrrolidin-1-yl)pyrimidine
4-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
3-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1H-indazole
(2S,4S,5R)-4-(cyclopropylcarbamoyl)-2-ethyl-5-(4-fluorophenyl)-1-methylpyrrolidine-2-carboxylic acid
1-(4-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]methanesulfonamide
2-[(E)-2-cyclohexylethenyl]-N,N-dimethylpyridine-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
5-acetyl-N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]thiophene-3-carboxamide
N-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-(adamantan-1-yl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(3-phenylpropyl)piperidin-4-yl)methanol
1-[(1-{6-[(2-methylprop-2-en-1-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-(1H-imidazol-1-yl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine-4-carboxylic acid
[7-(2-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclohexyl-4-[2-(4-fluorophenoxy)ethyl]piperazine
2-acetyl-8-(2-phenoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-oxo-5-phenoxy-1-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1,4-dihydropyridine-3-carboxylic acid
3-(2-hydroxyethyl)-N-(5-methoxy-2-methylphenyl)-4-(2-methylpropyl)piperazine-1-carboxamide
2-amino-N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-methyl-1,3-thiazole-5-carboxamide
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
7-fluoro-2-methyl-4-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]quinoline
N-(1-methoxypropan-2-yl)-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(1-benzyl-4-phenylpiperidine-4-carbonyl)pyrrolidin-3-amine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
({1-[(1-{furo[3,2-c]pyridin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)dimethylamine
5-propyl-1'-(pyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(2-hydroxypyridin-3-yl)methyl]amino}methyl)piperidin-2-one
5-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
N-(3-ethoxypropyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-N,N-dimethylfuran-2-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
N-[(3R,4S)-1-[(2-aminopyrimidin-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3,3-trifluoropropanamide
2-(4-fluorophenyl)-4-(6-methoxypyrimidin-4-yl)morpholine
4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-2-one
1-[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
N-(2-methoxy-5-methylphenyl)-2-[2-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
3-ethoxy-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
3-{[1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]methyl}benzamide
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide