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5-(3-phenylpropyl)-5-(piperidin-4-yl)-3-(1,3-thiazol-2-ylmethyl)imidazolidine-2,4-dione
5-(2-chlorophenyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylfuran-2-carboxamide
N-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
4-(4-fluoro-2-methylphenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
(4aS,8aS)-2-(5-fluoropyridin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
3-{[(2-hydroxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}-8-methyl-1,2-dihydroquinolin-2-one
2-({5-[1-(propan-2-yloxy)ethyl]-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
(3R,4R)-4-methyl-1-(2-methyl-1,3-benzoxazole-6-carbonyl)-3-(propan-2-yl)pyrrolidin-3-ol
(2R,6S)-2,6-dimethyl-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}morpholine
ethyl 2-{1-[4-(4-hydroxyphenyl)benzoyl]piperidin-2-yl}acetate
1-(2-methoxyethyl)-5-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrrolidine-3-carboxamide
N-({1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
5-methyl-3-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
1-(2-{[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]amino}pyrimidin-4-yl)piperidin-3-ol
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)acetamide
4-benzyl-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[3-(1H-pyrazol-1-yl)propyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-methyl-5-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(pyrazin-2-yl)propanamide
N-methyl-6-(1-methyl-1H-imidazol-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}pyridazin-3-amine
4-methyl-5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
4-(5-{[(pyridin-2-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
7-(cyclopropylmethyl)-2-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N-(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(furan-2-ylmethyl)-4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazine
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-N-phenylpropanamide
2-(morpholin-3-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{4-[(2-chloro-4,6-dimethoxyphenyl)methyl]morpholin-3-yl}acetic acid
5-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
{1-[3-(4-fluorophenoxy)propyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
2-methyl-6-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]pyrimidin-4-ol
3-[(3R,4S)-1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-(2-chlorophenoxy)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(pyridin-4-yl)acetamide
1-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)urea
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-4-cyclopentylpyrimidine
4-fluoro-N-(3-{4-[(oxolan-3-yl)amino]piperidin-1-yl}phenyl)benzene-1-sulfonamide
1-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]piperidine-4-carboxamide
2-[5-(1-ethyl-1H-pyrazol-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]acetamide
N-ethyl-2-{5-[morpholin-4-yl(phenyl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-[4-(hydroxymethyl)phenyl]ethan-1-one
5-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione