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8-cyclopropanecarbonyl-2-(3-methylfuran-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[6-(trifluoromethyl)pyridin-3-yl]-2,3-dihydro-1H-isoindole
3-[(3R,4S)-4-(dimethylamino)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]propan-1-ol
4-[(4-fluorophenyl)methyl]-1,3-bis(propan-2-yl)-1,4-diazepan-5-one
9-(5-chloro-2-fluorobenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N-(5-cyano-1,3-thiazol-2-yl)-3-[(diethylamino)methyl]benzamide
5-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-3-propylimidazolidine-2,4-dione
4-ethyl-1-methyl-3-{1-[2-(methylamino)pyridine-3-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1S,2R)-2-aminocyclobutyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(azepane-1-carbonyl)-5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
2-{[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
1-methyl-9-(prop-2-en-1-yl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(3-methoxypropyl)-3-{[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}benzamide
N-tert-butyl-5-methyl-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-acetyl-N-ethyl-2,4-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrrole-3-carboxamide
4-(1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1H-imidazol-2-yl)pyridine
14-(3-chloro-5-fluoro-4-methoxyphenyl)-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{[4-(2-chlorophenyl)-5-[(4-hydroxyphenyl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{4-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-(propan-2-yl)pyrimidine
1-(1-benzothiophen-2-ylmethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
5-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-3-(thiophen-2-yl)-1H-pyrazole
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
ethyl 4-{[5-(2H-1,3-benzodioxol-5-yl)-2-hydroxyphenyl]methyl}piperazine-1-carboxylate
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2,8-dimethyl-3-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
1-cyclopropyl-3-(1-propyl-1H-1,3-benzodiazol-5-yl)-1-(1,3-thiazol-2-ylmethyl)urea
2-amino-N-cyclobutyl-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-cyclohexyl-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
(1S,2R)-N1-methyl-N1-(3-phenylpropyl)-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
1-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-[(1S,2R)-2-phenylcyclopropyl]urea
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-3-ethoxypropanamide
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-[2-(pyrrolidine-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}adamantan-1-yl acetate
N-methyl-1-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidine-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-(1,4-dithiepan-6-yl)piperidin-3-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2,2,3,3-tetrafluoropropoxy)acetamide
2-(4-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
methyl 3-{[(2E)-3-(2-chlorophenyl)prop-2-enamido]methyl}-5-(furan-2-amido)benzoate
2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroisoquinolin-1-one
2-[(2-methoxyethyl)(methyl)amino]-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[2-(4-phenylpyrimidin-2-yl)ethyl]urea
(1R,3S)-7-(2,3-dimethyl-1H-indole-7-carbonyl)-3-[2-(dimethylamino)ethoxy]-7-azaspiro[3.5]nonan-1-ol
2-({[3-(dimethylamino)propyl]amino}methyl)-6-methylquinolin-4-ol
N-[4-(2-ethylbenzamido)phenyl]-5-methylfuran-2-carboxamide
2-(1-{1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-amine