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N-[(3-propyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-(1-{[(1-phenyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
3-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propanamide
3-(2-methylpropyl)-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1,2-oxazole-5-carboxamide
(2S)-2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-phenylpropan-2-amine
1-cyclobutanecarbonyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(dimethylamino)-2-(3-fluorophenyl)acetamide
2-(4-chlorophenyl)-4-[4-(prop-2-en-1-yl)benzoyl]morpholine
2-[(5-{2-amino-3-cyano-5H-chromeno[4,3-b]pyridin-4-yl}pyrimidin-2-yl)amino]acetic acid
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]propanamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
5-(3-methoxyphenyl)-2-(pyridin-4-yl)-4-[1-(thiophene-3-carbonyl)piperidin-4-yl]pyrimidine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
{1-[(4-methoxyphenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
2,5-dimethyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
1-(furan-3-ylmethyl)-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[1-(3,4-dimethylbenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
5-chloro-4-[4-({imidazo[1,2-a]pyridin-2-ylmethyl}amino)piperidin-1-yl]-6-methylpyrimidin-2-amine
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
methyl N-{2-oxo-2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]ethyl}carbamate
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
2-ethoxy-5-[2-(pyridin-2-yl)pyrimidin-4-yl]benzoic acid
N-{2-fluoro-5-[({[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}carbamoyl)amino]phenyl}acetamide
4-[4-(dimethylamino)azepane-1-carbonyl]-2-methoxyphenol
(3S,4S)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-methylpiperidine-3,4-diol
N,N-dimethyl-3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}benzamide
2-(2-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
[1-({[4-(ethylamino)pyrimidin-2-yl](methyl)amino}methyl)cyclobutyl]methanol
4-(azepan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxobutanamide
(3S,4S)-1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
2-({4-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-phenyl-4-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}piperazine
1-({1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
7-methyl-2-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1,5-dimethyl-4-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(1-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
N-methyl-5-(4-methylpiperazin-1-yl)-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{3-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]phenoxy}ethan-1-ol
3-methyl-1-phenyl-5-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-[4-(piperidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
N-butyl-1-(furan-2-ylmethyl)-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
7-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1-oxa-7-azaspiro[3.5]nonane
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}benzamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-methylphenoxymethyl)piperidine
1-ethyl-N-[2-(piperidin-1-yl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine