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N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-methyl-2-oxo-6-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-(3,5-dichlorophenyl)-1,2,4,5,10,11-hexaazatricyclo[7.3.0.02,6]dodeca-3,5,7,9,11-pentaene
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-9H-fluorene-9-carboxamide
N-[(3-chlorophenyl)methyl]-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
1-(2-methoxy-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
1-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
[(2,4-difluorophenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-[(3R,4S)-1-[(2-ethylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-ethyl-1H-pyrazole-5-carboxamide
N-(1,4-dioxan-2-ylmethyl)-N-methylisoquinoline-1-carboxamide
1-tert-butyl-4-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[2-(1,3-benzoxazol-2-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1'-(5-chloropyridin-2-yl)-5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(morpholin-4-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperidin-3-ol
4-{2-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]ethyl}benzene-1-sulfonamide
methyl 3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]benzoate
6-methyl-2-(thiomorpholin-4-ylmethyl)quinolin-4-ol
[(2S,6S)-4-{[4-(trifluoromethoxy)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(3-methylphenyl)piperidine-1-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methylbenzamide
5-(2,3-dimethoxyphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
6-(1-{[1-(propan-2-yl)-2,3-dihydro-1H-indol-5-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
(1R,3S)-3-methoxy-7-(2,4,5-trifluorobenzoyl)-7-azaspiro[3.5]nonan-1-ol
N-[2-(5-methyl-4-{[methyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})amino]methyl}-1,3-oxazol-2-yl)phenyl]methanesulfonamide
4-(3-methylphenyl)-3-(oxan-4-yl)-4H-1,2,4-triazole
2-amino-4-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-{2-[4-(4-methylphenyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
ethyl 1-[(3-hydroxy-4-methoxyphenyl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
methyl 3-(4-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)quinoline
3-[(4-fluorophenyl)methyl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2-oxazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-fluoro-5-sulfamoylbenzamide
(1R,2R,4R)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-methoxy-N-({5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
3-({1-[2-(4-chlorophenoxy)acetyl]pyrrolidin-3-yl}methyl)benzamide
3-[4-(1-hydroxy-3-methylbutyl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine
4-(4-methyl-1H-pyrazol-1-yl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidine-4-carboxylic acid
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{2-methyl-3-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]propyl}acetamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl]methanol
(1,4-dioxan-2-ylmethyl)(methyl)[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-(cyclopropylmethyl)-5-(methoxymethyl)-N-propyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-(3-methylpiperidin-1-yl)-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one