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N-(3-carbamoyl-4-fluorophenyl)-4-(2-methoxyphenoxy)piperidine-1-carboxamide
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
5-[(methylsulfanyl)methyl]-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[(2-methoxyphenyl)methyl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2-{4-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)morpholine
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
N-(1H-indol-4-ylmethyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-2-carboxamide
1-(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
7-methyl-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
N-[2-(1H-imidazol-4-yl)ethyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-4-(oxolan-2-ylmethyl)piperazine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(pyridin-4-yl)propyl]-1H-pyrazole-3-carboxamide
3-{[3-(2,5-dimethylfuran-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}benzonitrile
4-{[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]propan-1-one
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(piperidine-1-sulfonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,2-oxazolidin-4-ol
5-({methyl[(5-methylthiophen-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
3-(2-fluorophenyl)-5-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[1-(3-methylbut-2-en-1-yl)-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N-({2-[(3,4-dimethoxyphenyl)methyl]-6-oxo-1,6-dihydropyrimidin-4-yl}methyl)acetamide
1-benzyl-N,N-dimethyl-5-[(2-phenylethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(2-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-3-amine
1-(2-methoxyethyl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
4-(2-ethylphenyl)-6-methoxypyrimidin-2-amine
2-(adamantan-1-yl)-5-(4-hydroxypiperidine-1-carbonyl)pyrimidin-4-ol
[2-(2-methoxyphenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
ethyl 4-(3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperazine-1-carboxylate
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
5-cyclopropanecarbonyl-1'-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-benzyl-5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]-N-(2-methylpropyl)piperidine-3-carboxamide
4-{3-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]propyl}-1H-pyrazole
1-(ethanesulfonyl)-4-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazine
2-hydroxy-3-methyl-1-[6-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(2R,3R)-3-(dimethylamino)-N-(furan-2-ylmethyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
(2R)-2-{[3-(1H-imidazol-2-yl)phenyl]formamido}-4-methylpentanamide
6-[2-(4-methyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]-1H-indazole
(1S,5R)-3-{[3-(2-aminoethyl)phenyl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-acetyl-1H-1,3-benzodiazol-1-yl)-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
1-ethyl-3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]urea
7-(cyclopropylmethyl)-2-[(5-methylthiophen-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-(cyclohex-1-en-1-yl)acetyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(2S,4S)-N-(furan-3-ylmethyl)-4-(2-methoxybenzamido)-1-methylpyrrolidine-2-carboxamide
(4aR,7aS)-1-acetyl-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-({1-[2-(4-methoxyphenoxy)ethyl]piperidin-4-yl}methyl)pyrrolidin-2-one
6-[2-(trifluoromethyl)morpholine-4-carbonyl]quinoline