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1-methyl-2-[3-(2-methylphenyl)benzoyl]-1H-imidazole
5-(3-fluoro-4-methoxyphenyl)-1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-4-phenyl-1H-imidazole
1-[4-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)thiophen-2-yl]ethan-1-one
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-[(6-methylpyridin-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-hydroxy-3-methylbutyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
2,3-dimethyl-6-[4-(piperidin-1-yl)benzoyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
3-{4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-1H-pyrazole
{4-[(1-benzyl-1H-indol-6-yl)methyl]-1,4-oxazepan-6-yl}methanol
4-(piperidin-3-yl)-N-(2,2,2-trifluoroethyl)benzamide
4-{4-[(3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-(2-fluorophenyl)piperidin-4-ol
N-[2-(benzylsulfanyl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(3-methoxyphenyl)-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
4-(2-ethoxyphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]ethan-1-one
6-chloro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}pyridazin-3-amine
5-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-(4-methylphenyl)pyrimidin-5-yl}pyridin-2-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methylpyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
(3S,4S)-1-(4-methoxypyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
5-(1H-indol-1-ylmethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
N-{1-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
N-(3-ethoxypropyl)-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-(2,3-dihydro-1H-inden-2-yl)-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[2-(thiophen-2-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
5-(2-hydroxy-5-methoxybenzoyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(3-fluorophenyl)-8-methoxy-5-(quinoxalin-6-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine
1-{[5-(ethylsulfanyl)-1,3,4-oxadiazol-2-yl]methyl}-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
ethyl 2-[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-2-yl]acetate
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclobutanamine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
N-{2-[2-(3-chlorophenyl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
1-[1'-(3-fluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
6-methoxy-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-(4-fluorobenzenesulfonyl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
1-(1-propylpiperidin-4-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
8-cyclopropanecarbonyl-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 2-(4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)acetate
1-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
(1R,5S,6R,7S)-3-cyclopentyl-4-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[(3S,5S)-1-acetyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
2-(2-chloro-4-fluorophenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-(4-methylpiperazin-1-yl)-6-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-2-amine
N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-(thiophen-3-ylmethyl)benzamide
(2R,3R)-3-{[2-(pyridin-2-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3,3-dimethylbutan-1-one