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4-(1-{1-[2-(propan-2-ylsulfanyl)ethyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
4-[(2-chlorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidine-4-carboxylic acid
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-benzothiophene-5-carboxamide
methyl 1-[3-(furan-3-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]-4-(piperidin-1-yl)piperidine-4-carboxamide
1-{[1-(2-hydroxyethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,4-dihydroquinolin-4-one
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-amino-4-[(benzyloxy)methyl]-6-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-(2,6-difluorophenyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
6-(dimethylamino)-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
N,4-dimethyl-5-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-[(4-methylphenyl)methyl]-3-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanamide
N-cyclopropyl-1,6-dimethyl-2-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
(5-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(1-{2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carbonyl}pyrrolidin-3-yl)acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-ethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-pyrrole-2-carboxamide
3-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]pyridine
{4-[4-methoxy-3-(morpholin-4-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
2-benzyl-8-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
N-[1-(benzenesulfonyl)azepan-3-yl]-2-(3-methyl-1,2-oxazol-5-yl)acetamide
2-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
4-{[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}benzonitrile
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
3-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
6-methyl-2-{[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]amino}-3,4-dihydropyrimidin-4-one
3-[1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
6-methyl-2-{[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}pyridin-3-ol
N-[(3R,4R)-3-hydroxypiperidin-4-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
(3R,4R)-1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-4-(hydroxymethyl)piperidin-3-ol
1-(3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-1,2,4-triazole
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
4-methoxy-N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
3-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-N,N-dimethylaniline
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylacetamide
1-(4-methyl-2-{[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]amino}pyrimidin-5-yl)ethan-1-one
3-(piperidin-1-ylmethyl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}pyrrolidin-3-ol
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1-methyl-1H-pyrazol-4-yl)pyridine
5-(3-fluorophenoxymethyl)-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
2-ethyl-9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,2,3-thiadiazole
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-[4-(hydroxymethyl)phenyl]acetamide
N,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(morpholin-4-yl)ethyl]quinoline-4-carboxamide