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4-(2-methoxyethoxy)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(5-methylthiophen-2-yl)methyl](piperidin-3-ylmethyl)(pyridin-2-ylmethyl)amine
(1R,2R)-2-[5-(1H-imidazol-1-ylmethyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
4-[1-(2-fluorophenyl)piperidin-4-yl]-1,4-oxazepan-6-ol
5-[2-(benzenesulfonyl)ethyl]-1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazole
5-(1H-pyrazol-3-yl)-N-(pyridin-3-yl)furan-2-carboxamide
2-methyl-1-(2-{5-[3-(morpholin-4-yl)azetidine-1-carbonyl]thiophen-2-yl}pyrrolidin-1-yl)propan-1-one
5-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-(pyridin-2-yl)pyrimidine
1-methyl-2-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-indole
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
3-[2-(dimethylamino)ethyl]-1-(3-methylbutyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(isoquinolin-5-ylmethyl)({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
dimethyl({1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
1-(azepan-1-yl)-3-(3-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
2-{5-methyl-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-2-oxopiperazin-1-yl}benzonitrile
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(piperidin-1-yl)ethyl]amine
1-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2,6-difluoro-4-methoxybenzoyl)piperidine
5-chloro-2-{4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}pyrimidine
3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[2-(piperidin-1-ylmethyl)phenyl]urea
4-[7-(3-chloropyridin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
9-[(2,3-difluorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[4-(2H-1,3-benzodioxol-5-yl)phenyl]ethyl}acetamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-3-carboxamide
4-ethyl-1-methyl-3-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(naphthalen-2-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1,2,4-triazin-3-amine
2-[4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]-N-(2-fluoro-4-methylphenyl)acetamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-propoxypropan-1-one
7-(oxane-2-carbonyl)-N-(1,2-oxazol-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
3-(5-methylfuran-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
9-(5-hydroxypyrazine-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-chloro-4-fluoro-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-benzothiophene-2-carboxamide
2-(4-methyl-1H-pyrrole-2-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-(morpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N,3,5-trimethyl-N-[2-(oxan-4-yl)ethyl]-1-benzofuran-2-carboxamide
1-[(2-ethoxy-3-methoxyphenyl)methyl]-2-(furan-3-yl)-1H-imidazole
4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1-(2-methylphenyl)piperazin-2-one
1-(5-acetylthiophene-3-carbonyl)-4-[(2-chlorophenyl)methyl]-1,4-diazepan-5-one
1-(3-carbamoyl-6-methylpyridin-2-yl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-methyl-6-[2-(pyridin-4-yl)-1H-imidazol-1-yl]heptan-2-ol
5-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(propan-2-yl)propanamide
(3S,4R)-1-[3-(dimethylamino)benzoyl]-4-phenylpyrrolidine-3-carboxylic acid
3-(2-ethylphenoxy)-1-(oxolan-3-ylmethyl)azetidine
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(1H-indol-2-yl)pyridine-3-carbonitrile
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide