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2-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyridin-3-ol
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
(1R,5S,6S)-6-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
2-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-acetyl-N-[(1-benzylpyrrolidin-3-yl)methyl]benzamide
3-methyl-1-[(3-phenylphenyl)methyl]pyrrolidin-2-one
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5,6-dimethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-cyclopentylpyridin-2-amine
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]pyridin-2-amine
N-(2,2-difluoroethyl)-3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(oxan-4-yl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,4-diazepan-6-ol
1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(2-oxo-2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydroquinolin-2-one
N-(furan-2-ylmethyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine-4-carboxamide
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
(3aS,6aR)-5-(2-aminoacetyl)-3-[3-(4-methoxyphenyl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cycloheptanecarbonylpiperidine
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
N-{[4-(hydroxymethyl)phenyl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(oxan-4-ylmethyl)amino]methyl}piperidin-2-one
2-{[4-(2-methoxy-5-methylphenyl)-5-(piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
[(2S,6S)-11-methoxy-4-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
2-[methyl({4-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]phenyl})amino]ethan-1-ol
2-[methyl(pyridin-4-ylmethyl)amino]-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]ethan-1-one
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-5-methyl-2,1,3-benzothiadiazole-4-sulfonamide
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
2-oxo-2-(pyridin-3-yl)-N-[3-(pyridin-4-yl)propyl]acetamide
2-{1-[1-(oxan-4-yl)piperidine-4-carbonyl]pyrrolidin-2-yl}pyridine
3-{[5-(4-methoxy-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
4-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-methyl-3-[methyl({[4-(2-methylphenyl)phenyl]carbamoyl})amino]butanamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-cyclopropyl-5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3,4-oxadiazole
5-fluoro-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-1-methyl-1H-indole-2-carboxamide
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2-methyl-1-benzofuran-7-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-chloro-4-({1-[(2-chlorophenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
7-(2-methylphenyl)-4-(piperidin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-cyclobutanecarbonyl-1-phenylpiperazin-2-one
(3-{[1-(2-chloro-4,5-difluorobenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
3-(4-methoxyphenyl)-N-(thiolan-3-yl)propanamide
4-(3-chloropyridin-2-yl)-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
9-ethyl-1-methyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazine
1-(cyclohexylmethyl)-5-[(3-ethoxypropyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid