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5-hydroxy-N-(5-methyl-2-pentanamidophenyl)pyrazine-2-carboxamide
4,4,4-trifluoro-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butan-1-one
2-(3-methoxypropyl)-9-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
7-methoxy-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
8-[3-(dimethylamino)propanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
5-methoxy-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1H-indazole
(3S,4S)-1-(2-aminopyridine-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-cyclohexyl-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-(isoquinolin-5-ylmethyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-ethoxy-5-[2-(4-fluorophenoxymethyl)pyrimidin-4-yl]benzoic acid
7-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]propan-1-one
5-[4-(piperidin-1-ylmethyl)phenyl]-1,2-dihydropyridin-2-one
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
1-(cyclohexylmethyl)-5-[(furan-2-ylmethyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3R,4S)-1-(3-methylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(morpholin-4-yl)acetamide
1-(4-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-benzyl-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-(1,4-diazepan-1-yl)-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
(2E)-N-(2-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)but-2-enamide
benzyl N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamate
2-{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-1,4-diazepan-6-yl}acetic acid
2,7,8-trimethyl-4-(3-phenylpiperazine-1-carbonyl)quinoline
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[5-methoxy-2-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-methoxy-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
2-(2,3-dimethylphenyl)-2-[4-(morpholin-4-yl)piperidin-1-yl]acetic acid
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-(piperidine-1-carbonyl)pyridine
methyl (2S,4S)-1-(naphthalen-2-ylmethyl)-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
[(2,6-dimethoxyphenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
4-ethyl-1-methyl-3-{1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(4-chloro-1H-pyrazole-3-carbonyl)piperidin-4-yl]pyrrolidin-2-one
(1S,6R)-9-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonane
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
1-(4-methanesulfonylpiperazin-1-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]amino}pyridine-3-carboxamide
2-{4-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]morpholin-3-yl}-N-propylacetamide
7-(3-chlorophenyl)-4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
ethyl 4-(3-phenylpropyl)piperidine-4-carboxylate
1-(furan-2-yl)-2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}ethane-1,2-dione
N-(2-methoxyethyl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-(thiophen-2-ylmethyl)benzamide