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1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-methyl-N-[(7-methyl-1H-indol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)(2-methylpropyl)amine
(1R,3S)-7-[1-(3,4-difluorophenyl)piperidin-4-yl]-7-azaspiro[3.5]nonane-1,3-diol
N-({1-[2-(ethylsulfanyl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)acetamide
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
3-(1-methyl-1H-pyrazol-4-yl)-1-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[benzyl(methyl)amino]piperidin-1-yl}propan-1-one
2-[1-(3-methylbut-2-en-1-yl)-4-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
2-(2-ethoxyphenyl)-2-[4-(morpholine-4-carbonyl)piperidin-1-yl]acetic acid
methyl 5-(2-propyl-1,3-thiazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(4-phenylphenyl)-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-[4-(5-chloro-2-methoxyphenyl)phenyl]-2-methoxyacetamide
(4aR,8aR)-2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[4-(2-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
4-{4-[(4-ethylphenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(1-phenylpropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
1-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]pyrrolidine-3-carboxamide
2-methoxy-4-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenol
7-(1H-indole-7-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-N-(2-ethoxyphenyl)piperidine-1-carboxamide
2-ethyl-4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
1-(3,4-dimethoxyphenyl)-N-(4H-1,2,4-triazol-4-yl)cyclopentane-1-carboxamide
3-ethyl-8-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7,7-dimethyl-2-[1-(propan-2-yl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-methoxy-6-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-(3-chloro-4-fluorophenoxy)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
7-(3-chlorophenyl)-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[5-(4-ethenylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-4-methylpiperazine
methyl 2-(1-{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}-3-oxopiperazin-2-yl)acetate
1-[4-(cyclopropylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperazin-2-one
[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
5-(3-acetamidophenyl)-N-(pyridin-3-yl)furan-2-carboxamide
(4aR,7aS)-1-benzyl-4-[3-(dimethylamino)-2,2-dimethylpropyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-1,4-diazepan-6-yl]acetic acid
1-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
1-(2-methoxyphenyl)-3-(1-{1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
7,7-dimethyl-2-[2-(propan-2-yloxy)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-(1,2-oxazole-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-ethyl-6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
2-cyclopropanecarbonyl-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-9-hydroxy-4H-pyrido[1,2-a]pyrimidin-4-one
1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
2-{4-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]phenoxy}acetamide