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3-(4-{[3-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
1-(2-ethylpyridine-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N6-cyclopentyl-N5-methyl-N5-(oxan-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[2-(4-fluorobenzenesulfonyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-methyl-5-{4-[1-(piperidin-1-yl)ethyl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
4-ethyl-3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(6-methylpyridine-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({2-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
(3aS,6aR)-3-(pyridin-2-ylmethyl)-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(3aR,5S,6S,7aS)-2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
4-(3-hydroxy-3-methylbutyl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-{4-[(3-methoxypyrrolidin-1-yl)methyl]phenoxy}-1-(4-methylpiperidin-1-yl)ethan-1-one
2-[2-(adamantan-1-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-phenoxyacetamide
5-(pyrrolidin-1-yl)-3-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridazine
3-{[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]methyl}benzonitrile
2-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
(3S)-4-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethylmorpholine
3-(2-methanesulfonylacetamido)-4-(2-methylpiperidin-1-yl)benzamide
3,5-difluoro-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-2-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrazol-3-yl)pyridine
5-methyl-2-(5-methylthiophen-2-yl)-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1H-pyrrole-2-carboxamide
3-phenyl-N-[4-(4-{[2-(pyrazin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]propanamide
1-[(3-hydroxy-4-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
9-(3-fluoro-4-methylbenzoyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
(3aR,6aR)-2-cyclopentyl-5-[(2,3,4-trifluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-2-(1-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)acetamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-{[3-(furan-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
3-(4-methyl-1,4-diazepane-1-carbonyl)-N-[(3R)-piperidin-3-yl]benzene-1-sulfonamide
ethyl 4-{[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
2-{5-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1'-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamide
4-[(4-methyl-5-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
ethyl 4-[(3-methoxyphenyl)methyl]-1-[1-(methylsulfanyl)propan-2-yl]piperidine-4-carboxylate
2-[4-(2-methylphenoxy)piperidine-1-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-(2-phenylethyl)-7-[1-(trifluoromethyl)cyclopropanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(1S,5R)-3-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one