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N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-methoxy-2-phenylacetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carboxamide
N-(3,5-dimethoxyphenyl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)propanamide
(2S,4S)-4-(4-{2-[(4-ethylphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
4-fluorophenyl (7S,9aR)-7-(1H-indol-3-ylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
7-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-(4-cyano-2-fluorophenyl)-4-(1-hydroxy-3-phenylpropyl)piperidine-1-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]acetamide
2-(3,4-dimethoxyphenyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]acetamide
2-[3-oxo-9-(quinolin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(1H-pyrrole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(2-methoxyphenyl)-3-(2-methylpropyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
3-({2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
5-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(4-methoxyphenyl)-1-[3-(morpholin-4-yl)azetidin-1-yl]-3-phenylpropan-1-one
2-ethyl-9-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-1-[1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]butan-1-ol
1-(2-methyl-1-benzofuran-7-carbonyl)-4-[(1-methylpiperidin-4-yl)methyl]piperazine
5-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
5-(2-fluorophenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-hydroxy-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-methyl-1-propyl-N-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrazole-5-carboxamide
(1-{1-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
9-hydroxy-7-(5-methylthiophen-2-yl)-N-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
(4aS,7aR)-1-[(4-phenylphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(oxan-4-yl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
6-({[2-(morpholin-4-yl)pyridin-3-yl]methyl}amino)-N-propylpyridine-3-carboxamide
4-{5-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
4-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
5-[cyclohexyl(pyridin-3-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylic acid
N3-{1-[(3-chlorophenyl)amino]-2-methylpropan-2-yl}piperidine-1,3-dicarboxamide
methyl 4-[5-({4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2-[(4aR,7aS)-4-benzyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-(2-hydroxypropyl)-9-(3-phenoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(3-methoxyphenyl)methyl]-4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazin-2-one
5-(3-methoxyphenyl)-N-[2-(propane-2-sulfonyl)ethyl]furan-2-carboxamide
5-chloro-4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-1,3-dimethyl-1H-pyrazole
5-{[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}pentan-1-ol
7-(2-methyl-4-phenylpyrimidine-5-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl]propan-1-ol
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N-(4-{[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]methyl}phenyl)acetamide
(2R,3S,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)-N-(1,2,3-thiadiazol-5-yl)piperazine-1-carboxamide
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(1-methyl-1H-pyrrol-2-yl)methyl]piperidine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
5-(3,4-dimethylphenoxymethyl)-N-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide