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2-cyclopropyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5,6-dimethyl-2-({1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-2,3-dihydropyridazin-3-one
(3aR,6aS)-5-[2-hydroxy-3,5-bis(propan-2-yl)benzoyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
1-(1H-imidazol-2-ylmethyl)-5,5-diphenylpiperidin-2-one
N-[(4-methoxyphenyl)methyl]-3-(pyrrolidine-1-sulfonyl)-5-[(thiophen-2-ylmethyl)amino]benzamide
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1H-imidazol-2-ylmethyl)acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-methyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
3-[2-(diethylamino)-2-(furan-2-yl)ethyl]-1-(1H-indol-5-yl)urea
5-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
3-[2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
5-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
methyl[2-(morpholin-4-yl)ethyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-4-(pyridin-4-yl)-1,4-diazepane
2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyrrolidine-1-carboxamide
(4aS,8aR)-6-(pyrimidin-2-yl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
7-(cyclohexylmethyl)-3H,4H,5H-pyridazino[4,5-b]indol-4-one
3-(1H-imidazol-1-ylmethyl)-4-(4-methoxy-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-({[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amino)pyridine-3-carboxamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]imidazolidin-4-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-methoxy-4-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamido]phenyl}-3-methylbutanamide
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
3-ethyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1,2-oxazole-5-carboxamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine-4-carbonyl}morpholine
7-[4-(1,3-oxazol-5-yl)benzoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2,5-dimethyl-3-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrazine
4-methoxy-N-({1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyridine-4-carboxamide
2-methyl-6-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)phenol
2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1,3-benzoxazole
{6-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]pyridin-2-yl}methanol
(2S)-2-{[5-(3-acetylphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
1-(carbamoylmethyl)-N-(cyclohex-1-en-1-ylmethyl)piperidine-4-carboxamide
(4aS,8aR)-6-[2-(2-chloro-6-fluorophenyl)acetyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-[1-(propan-2-yl)piperidin-4-yl]-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
4-{2-methyl-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-2-yl}morpholine
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-(1-{1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
1-(methoxymethyl)-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]cyclopropan-1-amine
1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
(3S,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-methylpiperidine-3,4-diol
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-benzyl-3-ethyl-1-(2-methoxy-2-methylpropanoyl)-1,4-diazepan-5-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]cyclopropanecarboxamide
8-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]quinoline