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1-[2-(4-chlorophenyl)morpholin-4-yl]-2-hydroxyethan-1-one
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
3-(5-methylfuran-2-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
4-{4-[methyl(1,3-thiazol-2-ylmethyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
1-{4-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepan-1-yl}ethan-1-one
N-(1-cycloheptylpiperidin-3-yl)-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(1R,5S)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-methoxyacetyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
5-cyclopropanecarbonyl-1'-(2,6-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-cyclobutyl-N-[3-(1H-indazol-1-yl)propyl]-1,3,4-oxadiazol-2-amine
2-(5-acetylthiophen-3-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-(2-methoxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
(3R,4R)-4-(morpholin-4-yl)-1-(4-phenyl-1,3-thiazol-2-yl)piperidin-3-ol
5-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
methyl 2-({7-acetamido-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazol-5-yl}formamido)-4-(methylsulfanyl)butanoate
6-methyl-2-({[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}methyl)quinolin-4-ol
2-{5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-amino-4-(3-ethenylphenyl)-6-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
3-cyano-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)benzamide
3-{1-[2-(1H-imidazol-1-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
1-[({[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
2-(cyclopropylamino)-1-{4-[(2-fluorophenyl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(3S,5R)-5-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}pyrrolidin-3-ol
4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(pyridin-3-yl)benzamide
1-(furan-2-ylmethyl)-4-(3-methylphenoxy)piperidine
(1S,5R)-3-(1,3-thiazol-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
(1S,5R)-6-benzyl-3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-4-(pent-2-yn-1-yl)-1,4-diazepane-6-carboxylic acid
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
N,1-dimethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]azepane-2-carboxamide
1-[2-(2-methylphenyl)acetyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
2-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-tert-butyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
3,5,7-trimethyl-2-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]-1H-indole
4-(4-methanesulfonylphenyl)-3,5-dimethyl-1,2-oxazole
4-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-3-carbonyl)morpholine
methyl 4-{[7-oxo-4-(thiophene-2-carbonyl)-1,4-diazepan-1-yl]methyl}benzoate
4-(4-hydroxyphenyl)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
4'-[(dimethyl-1,2-oxazol-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3aR,6aR)-2-acetyl-5-[2-(3-ethoxyphenoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid