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1-(carbamoylmethyl)-N-[3-(2,4-dimethylphenoxy)propyl]-N-methylpiperidine-3-carboxamide
3-(5-methylthiophen-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-5-carboxamide
3-(oxan-4-yl)-5-[5-(1H-pyrazol-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazole
2-[(1S,5R)-6-{[2-(2-hydroxyethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(butan-2-yl)[(2-propylpyrimidin-5-yl)methyl](pyridin-4-ylmethyl)amine
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-methyl-N-(quinoxalin-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
4-(1-butyl-1H-imidazol-2-yl)-1-(propane-2-sulfonyl)piperidine
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-benzyl-1H-pyrazole-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylsulfamoyl)ethyl]propanamide
1-methyl-3-{[1-(oxolan-3-ylmethyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-methylphenyl)methyl]-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-{[(5-methylthiophen-2-yl)methyl]amino}benzamide
1-(oxan-4-yl)-4-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidine
8-(4-methyl-1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-fluoro-N-({3-methyl-7-[(4-oxo-4H-chromen-3-yl)methyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
3-(3-chloro-1,2-oxazol-5-yl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
(2R,6R)-4-[(2-aminopyridin-3-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
5-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
(4aS,8aR)-6-[(5-methylfuran-2-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(2-methylphenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
N-(2-methoxyethyl)-2-(2-methoxyphenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
methyl 3-{[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)carbamoyl}propanoate
5,7-dimethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
7-(3-chlorophenyl)-4-(furan-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(cyclopropylmethyl)-1-(2-hydroxy-5-methylbenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(3aS,7aR)-2-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
4-(4-chlorophenoxy)-1-(3-methylpyridine-2-carbonyl)piperidine-4-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
(3aR,6aS)-5-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-2-{4-[2-(2-methoxyphenyl)-1H-imidazol-1-yl]phenyl}acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2,4-dimethylpyrimidine-5-carboxamide
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2-(2,3,4-trifluorophenyl)acetamide
N-[(3R,4S)-1-[(4-methoxypyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]cyclopropanesulfonamide
[2-({1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]piperidin-4-yl}oxy)ethyl]dimethylamine
8-[(3-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
4-[(2-methylphenyl)sulfanyl]-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
6-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-1,4-oxazepan-6-ol
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
[(1-{1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl](methyl)amine
1-methyl-3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[3-(pyridin-2-yl)-1,2-oxazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one