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(3R)-3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-[2-({[2-(diethylamino)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-(2,6-dimethoxypyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-4-cyclobutyl-3-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidin-4-ol
N1-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-N3-methylpyrrolidine-1,3-dicarboxamide
4-(pyrrolidin-1-ylmethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-ol
3-[(3R,4S)-4-(dimethylamino)-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl]propanoic acid
1-{3-[4-(6-methylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-1,2,3-benzotriazole
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-(1H-imidazol-2-yl)-1-[4-(1H-pyrazol-4-yl)phenyl]-1H-imidazole
4-[5-(2-chlorophenyl)furan-2-carbonyl]-3-(2-hydroxyethyl)piperazin-2-one
3-(4-phenyl-1H-pyrazol-5-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
(2R)-2-amino-N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-methylpentanamide
2-[1-cyclopentyl-4-(isoquinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[3-({[2-(morpholin-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-cyclobutyl-4-methylpyrrolidin-3-ol
2-[(4-chlorophenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-5-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(6-cyclopropylpyrimidin-4-yl)phenyl]methyl}morpholine
N-(2,6-dimethylphenyl)-4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N4-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(6-phenoxypyridin-3-yl)piperidine-1-carboxamide
(1R,5S,6R)-3-cyclopropanecarbonyl-6-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-cyclohexyl-3-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)urea
3-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(2,3-dimethoxy-5-methylphenyl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
3-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-{2-[(2-benzyl-1,3-thiazol-4-yl)formamido]ethyl}pyridine-3-carboxamide
methyl 4-oxo-4-[3-(2-{[4-(trifluoromethyl)phenyl]carbamoyl}ethyl)piperidin-1-yl]butanoate
4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
1-[3-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-1-yl]ethan-1-one
(2S,4S)-4-[4-({[(4-cyanophenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-[(2-methoxyphenyl)methyl]-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-propylacetamide
N-methyl-N-[3-(phenylsulfanyl)propyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
(1R,6S)-9-methyl-3-[5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
N-[2-(3-methylthiophen-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-(4-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)-1H-1,2,4-triazole
5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-cyclopentyl-1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-[(3-fluorophenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
1-(3-methoxypropyl)-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[2-(3,4-difluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N'-(3-chlorophenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pentanediamide
N-{2-[(2-chlorophenyl)formamido]ethyl}-1-(2-methoxyacetyl)piperidine-3-carboxamide
2-benzyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1,3-thiazole-4-carboxamide
N-(3,4-dimethylphenyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
3-{imidazo[1,2-a]pyridin-2-yl}-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
2-(3-methoxypropyl)-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one