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3-benzyl-1-(3-methoxypropyl)-8-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-oxo-2-phenylacetamide
3-hydroxy-3-({[2-oxo-2-(piperazin-1-yl)ethyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
1-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
2-({4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-ethoxyphenol
4-chloro-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(oxolane-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
5-(3-fluorophenoxymethyl)-N-(3-hydroxy-2,2-dimethylpropyl)-1H-pyrazole-3-carboxamide
1-(1H-indazol-6-yl)-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperazin-2-one
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}morpholine
N,N-dimethyl-4-({2-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)oxan-4-amine
6-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyrazine-2-carboxamide
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol
1-{2-[1-(3-phenylpropyl)-1,2,5,6-tetrahydropyridin-3-yl]piperidin-1-yl}ethan-1-one
4-[7-(1H-pyrazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
(3S,5R)-5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
(1r,4r)-4-[({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]cyclohexan-1-ol
1-{2-[1-(3-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
2-[(1-propyl-1H-pyrazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[ethyl(2-methoxyethyl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
2-[3-({[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
9-[2-(4-fluorophenoxy)ethyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(4-chlorophenyl)-2-(2-methoxypropan-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]propan-1-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-(1H-indazol-1-yl)propyl]acetamide
(3S,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-N-[(4-methylphenyl)methyl]propanamide
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
1-[3-(4-chlorophenyl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-(carbamoylmethyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]piperidine-4-carboxamide
8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]cyclopentanecarboxamide
1-{2-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}pyrrolidin-2-one
ethyl 4-{[(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)carbamoyl]amino}piperidine-1-carboxylate
(1S,9S)-11-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2,4-dimethylpyrimidine
4-(1H-imidazole-5-carbonyl)-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(3-methoxyphenyl)methyl]-1,3-oxazole-4-carboxamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-(4-hydroxy-2-methylphenyl)pyridine-3-carbonitrile
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N,1,7-trimethyl-1H-indole-2-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-ethoxynaphthalen-1-yl)-1-ethyl-1H,4H-pyrazolo[3,4-d]imidazole
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2-methylpropyl)piperidine-4-carboxamide
3-(pyridin-3-yl)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
1-(azocan-1-yl)-3-(4-{[(2-hydroxyethyl)(propan-2-yl)amino]methyl}-2-methoxyphenoxy)propan-2-ol