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2-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
1-(carbamoylmethyl)-N-[2-(5-methoxy-1H-indol-3-yl)ethyl]piperidine-4-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propan-1-one
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[4-(1H-pyrazol-1-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[4-(5-cyclopropaneamido-1H-pyrazol-1-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(3S,4R)-1-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-4-phenylpyrrolidine-3-carboxylic acid
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(pyridin-3-yloxy)piperidin-1-yl]ethan-1-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-(7-chloro-9-oxo-9H-fluorene-1-carbonyl)-4-(cyclopropylmethyl)-1,4-diazepan-5-one
4-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
(furan-2-ylmethyl)[(6-methoxypyridin-3-yl)methyl](prop-2-en-1-yl)amine
N-(3-methylbutyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
8-fluoro-N-[3-(methylsulfanyl)propyl]quinoline-2-carboxamide
2-{4-[1-(furan-3-ylmethyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-[(4-methylphenyl)methyl]piperidin-4-ol
5-methyl-1-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(4aR,8aS)-1-[(3,4-dimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-6-yl]-2-phenylethan-1-one
2-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(4-fluoro-3-methylphenyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)urea
1-cyclopentyl-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}pyrrolidin-2-one
6-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2-methyl-1,3-benzoxazole
1-(4-ethoxyphenyl)-3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]urea
3-(4-hydroxyphenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
(1R,9S)-5-amino-12-methyl-3-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-methyl-N-[2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]propanamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-2-methyl-6-propylpyrimidine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-ol
3-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
3-{3-[(2-methoxyphenyl)methyl]-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
6-cyclopropyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-4-amine
3-{[4-(cyclobutylmethyl)piperazin-1-yl]methyl}-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
4-methyl-5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrimidin-2-amine
4-{[5-(2,3-dihydro-1-benzofuran-7-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
3-[2-(4-fluorophenyl)piperidine-1-carbonyl]pyridine
N-[(4-acetylmorpholin-2-yl)methyl]-5-propylthiophene-3-carboxamide
6-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[4-({[1-(2-methylphenoxy)propan-2-yl]carbamoyl}methoxy)phenyl]propanamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-2-sulfonyl)piperidine
N-methyl-N-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}oxan-4-amine
5-(3-fluorophenyl)-3-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-1,2,4-triazine
N-[(3R,4S)-4-(propan-2-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-yl]oxane-4-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
5-benzoyl-N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-2-oxoethyl}-1-methylurea
4-{1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid