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N-benzyl[(6-fluoropyridin-3-yl)amino]sulfonamide
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]-N-(4-methylphenyl)propanamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]benzamide
3-[4-(3-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
N-ethyl-6-methyl-5-{5-[2-(methylamino)pyridin-3-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-[2-(3-fluorophenyl)ethyl]-4-[4-(furan-3-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(4aR,8aR)-7-[(4-acetamidophenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
[(4-methyl-1H-imidazol-5-yl)methyl](propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1-methylazepane-2-carboxamide
3-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1-(4-methylphenyl)urea
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-cyclopentyl-N-methyl-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4,4,4-trifluoro-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
1-[(3-fluoro-2-methoxyphenyl)methyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
1'-(3-methoxybenzoyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[3-(2-chlorophenoxy)propyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1H-1,2,3-triazole
5-{4-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(2R,3R)-1'-[(3,5-dimethylphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N,N-dimethyl-2-[4-(2-methylphenoxy)piperidine-1-carbonyl]aniline
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(1-methyl-3-phenyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-methyl-2-(naphthalen-1-yloxy)propan-1-one
N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]furan-2-carboxamide
3-(1-ethyl-1H-imidazol-2-yl)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
ethyl 2-(1-{2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamido}cyclohexyl)acetate
methyl 2-{4-[2-amino-3-cyano-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridin-4-yl]phenoxy}acetate
N-[3-(2-ethylphenoxy)propyl]-N,6-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-methyl-1-oxobutan-2-yl)acetamide
2-{[3-(3-{furo[3,2-c]pyridin-4-yl}phenyl)-1H-pyrazol-1-yl]methyl}-3-methylpyridine
2-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine-3-carbonitrile
2-(4-{[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]methyl}phenoxy)acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-2-ethylpyrimidine-5-carboxamide
[1-(5-{[(2,3-difluorophenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
5-methyl-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
N-methyl-N-(oxolan-2-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
diethyl({[2-ethyl-5-(3-propylmorpholine-4-carbonyl)furan-3-yl]methyl})amine
6-{[(4,6-dimethylpyridin-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2,6-dimethylpyridine-4-carboxamide
4-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
N3,N5-dimethyl-4-oxo-1-(3-phenylpropyl)-N3-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(3S,4R)-N-benzyl-3-acetamido-4-(4-methoxyphenyl)pyrrolidine-1-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amine