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2-(4-fluorophenyl)-4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}morpholine
2-(pyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
ethyl 2-{1-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]piperidin-2-yl}acetate
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide
5-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(2S)-2-amino-3-(4-hydroxyphenyl)-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
methyl(pyrazin-2-ylmethyl)[2-(quinolin-4-yloxy)hex-5-en-1-yl]amine
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-4-(4-methoxyphenoxy)piperidine
9-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(4-methylpyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
1-ethyl-4-[4-(4-methylphenoxy)piperidine-1-carbonyl]pyrrolidin-2-one
N-(2,2-difluoroethyl)-4-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
4-(benzyloxy)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]butan-1-one
7-(cyclopropylmethyl)-2-(3-ethyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(2S,4R,6R)-2-{2-phenylimidazo[1,2-a]pyrimidin-3-yl}-6-(propan-2-yl)oxan-4-yl]acetamide
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-[3-(trifluoromethyl)phenyl]acetamide
N-(1-methyl-2-oxopyrrolidin-3-yl)-4-(thiophen-2-yl)butanamide
(2S)-N2-[2-(2-fluorophenoxy)ethyl]-N2-(2-methoxyethyl)pyrrolidine-1,2-dicarboxamide
3-(2-methoxyphenyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazine
1-(2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(3R,4S)-4-propyl-1-(thiophene-3-carbonyl)pyrrolidin-3-amine
(4aR,8aS)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-(pyridin-4-yl)ethan-1-ol
2-{1-cyclopentyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-(furan-2-ylmethyl)-7-(pyrazine-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[4-(5-chlorothiophene-2-carbonyl)morpholin-3-yl]-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]acetamide
4-(2-chlorobenzenesulfonyl)-9-[2-(1-methylpyrrolidin-2-yl)ethoxy]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(cyclohexylmethyl)-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
2-{1-methyl-5-[4-(morpholin-4-yl)phenyl]-1H-1,2,4-triazol-3-yl}acetamide
(1R,3S)-3-(2-aminoethoxy)-7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
ethyl 1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{[methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})amino]methyl}benzoic acid
2-[2-(methoxymethyl)pyrimidin-5-yl]-1H-1,3-benzodiazole-6-carboxylic acid
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]acetamide
(1R,5S,6S)-6-({4-[2-(4-chloro-2-methylphenoxy)ethyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
[(6-methylpyridin-2-yl)methyl](oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
6-methyl-2-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
N-[(3-methoxyphenyl)methyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-2-methylpropanamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-phenyl-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butane-1,2-dione