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1-(2-cyclohexylethyl)-3-hydroxy-3-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)piperidin-2-one
N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-fluoro-2-[(3-propoxypiperidin-1-yl)methyl]quinolin-4-ol
3-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-indazole
[(2S,6S)-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-benzyl-N-ethyl-5-(4-hydroxypiperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
(1S,2S,9S)-N-[4-(methylsulfanyl)phenyl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
N-[(3R,4R)-3-hydroxy-1-[2-(methylsulfanyl)benzoyl]piperidin-4-yl]pyridine-4-carboxamide
1-[(3S)-3-aminopiperidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
8-chloro-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-[(1S,5R)-6-[(2-chloro-6-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
7-{2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-oxoethoxy}-4,8-dimethyl-2H-chromen-2-one
N-cyclopentyl-4-(pyrimidin-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(2-hydroxyethyl)piperazin-2-one
2-{[4-(3-oxo-3,4-dihydropyrazin-2-yl)piperazin-1-yl]methyl}benzoic acid
(2S,4R)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-(furan-2-amido)pyrrolidine-2-carboxamide
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(1,3-thiazol-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
(3R,7S,8aS)-3-(2-methylpropyl)-7-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
(2E)-N-{[7-(2,3-dihydro-1H-inden-2-yl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
2,3-dimethyl-6-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
(2R,3R)-3-amino-1'-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[methyl(5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]ethan-1-ol
N-[2-(morpholin-4-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-tert-butyl-3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carboxamide
N-methyl-2-(2-phenylethyl)-N-(thiophen-2-ylmethyl)-1,3-benzoxazole-5-carboxamide
(2R)-2-amino-3-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}butanamide
4-(1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
2-({[5-(3,4-dimethylpiperazine-1-carbonyl)furan-2-yl]methyl}sulfanyl)pyrimidine
4-{4-[(cyclopent-3-en-1-yl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}pyrrolidin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
2-{2-[cyclopentyl(methyl)amino]ethyl}-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{2-chloro-4-[(2-methoxyethyl)carbamoyl]phenoxy}-N-(propan-2-yl)piperidine-1-carboxamide
3-[(dimethylamino)methyl]-1-(2-methyl-1-benzofuran-7-carbonyl)pyrrolidin-3-ol
[(3R,4R)-1-(4-chloro-1H-pyrazole-3-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
N-({8-[2-(2,4,6-trifluorophenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide
N-(5-methylpyridin-2-yl)-2-{3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}acetamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-[4-(thiophen-2-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-(3,5-dimethylphenyl)-2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoacetamide
1-(3-methoxybenzoyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)piperazine
2-methyl-9-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(4aS,7aR)-1-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-{6-methyl-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
N-(2-fluorophenyl)-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
N,1-dimethyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine