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6-methyl-5-[5-(5-phenyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(2S,4R)-1-[(2-chlorophenyl)methyl]-4-{[(3-methoxyphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(5-methylfuran-2-yl)methyl]-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(4,5-dimethylthiophen-2-yl)methyl]-4-[6-(propan-2-yl)pyridin-2-yl]piperazine
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(oxane-4-carbonyl)-1,4-diazepan-2-one
(3R,4S)-1-(2-methoxyethyl)-N,N-dimethyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
5-chloro-6-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]pyridine-3-carboxylic acid
4-({3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-cyclooctyl-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
4-(3-hydroxypyridine-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(propan-2-yloxy)ethyl]benzamide
8-{[3-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
4-({4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(pyridin-4-yl)ethyl]benzamide
4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(pyridin-4-yl)ethan-1-one
4-(4-cyclohexylpiperazine-1-carbonyl)-6-ethyl-1,2-dihydropyridin-2-one
methyl({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-4-phenylpiperazine
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-1-(pyrimidin-2-yl)piperidine-4-carboxamide
2,3-dimethyl-5-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-indole
7-(cyclopropylmethyl)-2-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-methoxyethyl)-2-[methyl(pyridin-3-ylmethyl)amino]-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-amine
N-methyl-6-{[2-(pyridin-3-yl)ethyl]amino}-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
N-{2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}cyclopropanecarboxamide
N-{2-[4-(4-methyl-1,4-diazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-(naphthalen-1-yl)acetamide
(3S,4R)-3-benzyl-4-methyl-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
N-[2-(5-methyl-4-{[methyl(pyridin-2-ylmethyl)amino]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-3-carboxamide
[1-(3,4-dimethoxyphenyl)propyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-(1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]phenol
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(oxolan-2-ylmethoxy)acetamide
2-[4-(2-hydroxybutyl)-2-oxopiperazin-1-yl]benzonitrile
5-{[({3-[2-(4-cyclobutanecarbonylpiperazin-1-yl)ethoxy]phenyl}methyl)(methyl)amino]methyl}pyrrolidin-2-one
N-({5-[(4-propoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1,3-dimethyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-fluoro-N-[2-(2-hydroxyethoxy)ethyl]-3-methyl-1H-indole-2-carboxamide
2-amino-8-[2-(3-methylphenyl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
(3R,4R)-3,4-dimethyl-1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-ol
1-(2-{1-[(5-fluoro-2-methylphenyl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}piperidin-1-yl)ethan-1-one