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4-(piperidin-3-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
4-[(1s,4s)-4-aminocyclohexyl]-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(8-methoxyquinolin-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-methyl-6-(pyridin-3-yl)-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3,4-dimethylphenyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
2-(2-methyl-1H-pyrrole-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
methyl 8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-methylbutoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
2-(3-{[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-methylfuran-3-carboxamide
N-(4-methyl-3-propanamidophenyl)-4-(pyridin-3-yl)piperazine-1-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1-benzofuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
2-({4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
8-{[2-(2-fluorophenyl)ethyl]carbamoyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
3,7-dimethyl-2-(1H-pyrazol-4-yl)quinoline
N-cyclopropyl-3-{5-[(2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-(3-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenyl)ethan-1-one
5-chloro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-1,2,4-triazole-3-carboxamide
ethyl 3,5-dimethyl-4-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]carbamoyl}-1H-pyrrole-2-carboxylate
7-acetamido-N-(oxolan-3-yl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-{1-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
3-(propan-2-yl)-5-({2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-benzyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methylpiperidine-3-carboxamide
N-(pyridin-2-ylmethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-sulfamoylbutanamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
3-(1-methyl-1H-pyrazol-5-yl)-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}propanamide
2-[3-(2,6-dimethylphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
1-(3-aminoazepan-1-yl)-4-(2,4,5-trimethoxyphenyl)butane-1,4-dione
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-N'-(2-methylphenyl)propanediamide
8-[5-(1H-imidazol-1-ylmethyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]quinoline
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
2-{[4-(2,4-difluorophenyl)-5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[3-(2-methylphenyl)piperidin-1-yl]propan-1-one
2-ethyl-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(3-methoxyphenoxy)propan-2-ol
3-(azocan-1-yl)-N-(1H-indol-2-ylmethyl)propanamide
2-methyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}thieno[2,3-d]pyrimidin-4-amine
4-({1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-3-yl}methyl)benzoic acid
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
7-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one