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6-[3-cyclopropyl-1-(2,5-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-2,3-dihydropyridazin-3-one
7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}quinoline
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(morpholine-4-carbonyl)piperidin-1-yl]propan-1-one
5-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3-chloro-1,2-dihydropyridin-2-one
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(4-methylpiperazin-1-yl)-2-(3-phenylpropyl)-2,3-dihydropyridazin-3-one
{1-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]cyclopropyl}methanol
N-(1-ethyl-1H-pyrazol-4-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carboxamide
(3S,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(azocan-1-yl)-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)propanamide
8-[2-(3-chloro-2,6-difluorophenyl)acetyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
1-methyl-N-[3-(4-methylpiperazin-1-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-(cyclohexylmethyl)-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-(3,4-difluorophenyl)-5-oxopyrrolidin-3-yl]-N,5-dimethyl-1H-imidazole-4-carboxamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]urea
(3R,4R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
(3S,5R)-N5-(2,3-dihydro-1H-inden-5-yl)-1-(1H-indol-3-ylmethyl)-N3,N3-dimethylpiperidine-3,5-dicarboxamide
2-methyl-6-[4-(pyrrolidine-1-sulfonyl)phenyl]-2,3-dihydropyridazin-3-one
6-(2,5-dimethoxyphenyl)-N,N-dimethylpyrimidin-4-amine
7-methyl-4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
2-[3-(furan-2-yl)propanoyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
4-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-methoxypyridine-3-carbonitrile
2-({[(3R,4R)-1-(4,6-dimethylpyridine-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-(2-hydroxy-3-methoxypropyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-methyl-1-(4-{5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
1-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-cyclopropyl-5-(4-phenylpiperidine-1-carbonyl)piperidin-2-one
3-amino-3-(3,4-dimethoxyphenyl)-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-1-yl)butanamide
3-methoxy-1-{2-[3-(3-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
ethyl 1-(1-methyl-1H-pyrazole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(pyrrolidin-1-yl)ethyl]piperazine
N-methyl-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-{[(2-chlorophenyl)methyl]sulfanyl}acetamide
3-(furan-2-ylmethyl)-1-[1-(4-methoxybenzoyl)azepan-3-yl]urea
3-{2-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-(1H-indazol-5-yl)-1-[(4-methanesulfonylmorpholin-2-yl)methyl]urea
N-ethyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
7-(3-methoxypropyl)-2-[(1-methyl-1H-indol-6-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-(1,4-dioxane-2-carbonyl)-2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine