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N-[(3-methylpyridin-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-chloro-4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
6-ethyl-2-methyl-N-{3-[(pyridin-3-yl)amino]propyl}quinoline-4-carboxamide
N-methyl-5-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
2-(azocan-1-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-benzyl-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[2-(2-hydroxyphenyl)acetyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-(1H-1,3-benzodiazol-1-yl)-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
2-[(4-chlorophenyl)methyl]-8-[(2S)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
5-oxo-1-(prop-2-en-1-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyrimidin-2-amine
2,6-dimethoxy-4-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)phenol
1'-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(2-ethylpiperidin-1-yl)propan-1-one
6-{[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]amino}-N,N-dimethylpyrazine-2-carboxamide
2-[4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
N-butyl-N-methyl-3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
methyl 1-{2-hydroxy-3-[3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-cyclopentyl-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-methylthiophen-2-yl)methyl]propanamide
2-(pyridine-4-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-(2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}benzoic acid
4-(3-methyl-1H-pyrazole-4-carbonyl)-2-(3-phenylpropyl)morpholine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
6-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(1R,9aR)-N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-octahydro-1H-quinolizine-1-carboxamide
2-(3,4-dichlorophenyl)-4-[1-(methoxymethyl)cyclobutanecarbonyl]morpholine
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
(1R,3S)-3-methoxy-7-(4-methoxy-3-methylbenzoyl)-7-azaspiro[3.5]nonan-1-ol
[(3R,4R)-1-(1,6-dimethyl-1H-indole-2-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N,2,3,5-tetramethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[2-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1,2-benzothiazol-3-one
2-chloro-N-{2-[(5-methyl-1,3-oxazol-4-yl)formamido]ethyl}benzamide
3-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[2-(1H-pyrazol-1-yl)phenyl]urea
4-chloro-3-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-methyl-1H-indazole
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
N'-(2-ethoxyphenyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanediamide
4-[(1S)-1-cyclohexylethyl]-3-(3-hydroxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-ethyl-5-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,4-triazole
1-[(2-chlorophenyl)methyl]-4-(4-hydroxy-3-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-cyclopentanecarbonyl-N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(2-fluorophenyl)-3,4-dihydropyrimidin-4-one
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[3-(morpholin-4-yl)propyl]piperidine-3-carboxamide
5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide