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(9aR)-2-methyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-butyl-1H-imidazol-4-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
N-[2-(2-methyl-4-oxopentanoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
3-methoxy-1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
7-[(3-methylphenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
2-(3-methoxyphenoxymethyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-4-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(2-methylbenzenesulfonyl)-decahydro-1,6-naphthyridin-2-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}pent-4-enamide
4-methyl-6-(4-{[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyridin-4-yl)ethan-1-ol
1-ethyl-3-[3-(pyridin-3-yl)propyl]-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-benzothiophene-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-phenylacetyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]isoquinoline-1-carboxamide
methyl (2S,4S)-4-(1,2,5-thiadiazole-3-amido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
2-({[(5-methoxy-1H-indazol-3-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
methyl (2R,4S)-1-(2-ethoxy-2-oxoethyl)-4-hydroxypiperidine-2-carboxylate
2-[(dimethylcarbamoyl)amino]-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]acetamide
[(3R,4R)-1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-cyclopropyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
2-ethyl-7-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
8-[5-(3-chloropyridin-4-yl)-3-methyl-1H-1,2,4-triazol-1-yl]quinoline
(2S,4S)-4-amino-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
3-(benzylsulfanyl)-1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]propan-1-one
5-methyl-N-[(1-phenylcyclopentyl)methyl]-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyrimidin-2-amine
(3R,4R)-4-(azepan-1-yl)-1-[(4-hydroxyphenyl)methyl]piperidin-3-ol
3-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-1-methyl-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}urea
1'-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
1-[2-chloro-5-(1H-pyrazol-1-yl)benzoyl]-3-phenylpiperazine
(3S,7S,8aS)-7-({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}amino)-3-[(4-methoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propyl]pyridin-3-amine
(2S,4S)-4-{[(2-chlorophenyl)methyl]amino}-1-{[4-(diethylamino)phenyl]methyl}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
ethyl 5-(1H-indazole-3-carbonyl)-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-methyl-3-(3-phenylpiperazine-1-carbonyl)-1,2-dihydroquinolin-2-one
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(propan-2-yl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-N-propylthiophene-2-carboxamide
ethyl 1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
8-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-4-ylmethyl)piperidine
2-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]pyridine-4-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyridine-3-carboxamide
5-(4-cyclohexylphenyl)-3-(3-methoxypiperidin-1-yl)-1,2,4-triazine
3-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
(1S,5R)-6-methyl-3-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one