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(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-({2-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
8-fluoro-2-[3-(morpholin-4-yl)azetidine-1-carbonyl]quinoline
ethyl 1-methanesulfonyl-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-ethylbutanamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
3-cyclohexyl-4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
3-{2-[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}-1,3-oxazinan-2-one
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(oxan-2-ylmethyl)amine
3-({[(3-chlorophenyl)methyl]amino}methyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-4H-chromen-4-one
5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
3-methyl-1-propyl-4-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
(3S,4R)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-benzyl-5-[(R)-methoxy(phenyl)methyl]-1H-1,2,4-triazole
3-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)piperidin-3-ol
4-[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N'-(5-chloro-2-methylphenyl)propanediamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
(1S,5R)-6-benzyl-3-(9H-purin-6-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxy-5-methylphenyl)-2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetamide
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-ethyl-3-methylpiperazin-2-one
5-chloro-3-ethyl-1-methyl-4-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-pyrazole
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methyl-1H-pyrrole-3-carboxamide
1-(3-chlorophenyl)-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-methylpiperazin-2-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2,5-difluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclopentyl-N-[(3R,4S)-4-cyclopropyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(1-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}piperidin-4-yl)propanamide
3-(1H-imidazol-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide
3-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(1H-indol-3-yl)ethyl]-3-methoxy-1,2-dihydropyridin-2-one
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}morpholine-4-sulfonamide
4-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
1-(2-methylpropyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
4-ethyl-3-{[1-(quinolin-4-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl][(3-methylthiophen-2-yl)methyl]amine
2-({2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)-3,4-dihydroquinazolin-4-one
N-(1-propyl-1H-pyrazol-5-yl)-2-[4-(1,3-thiazol-2-yl)-1H-pyrazol-1-yl]acetamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylbutan-1-one
(4aS,7aR)-1-(5-hydroxypyrazine-2-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3-{5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-methyl-2-[2-(2-methylpyrrolidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]propanoic acid
1-{3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}azepan-2-one
1-(furan-2-carbonyl)-N-(4-methoxy-4-methylpentan-2-yl)piperidin-4-amine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-yl)ethan-1-one