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1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-1-[4-(pyridin-4-yl)piperidin-1-yl]butan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperazin-2-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
5-(2-methoxy-5-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
(1R,3S)-7-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}-7-azaspiro[3.5]nonane-1,3-diol
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-4-hydroxy-2-(3-methylphenyl)pyrimidine-5-carboxamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-[1-(cyclohexylmethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
5-cyano-6-(3,5-dimethoxyphenyl)-2-methylpyridine-3-carboxylic acid
5-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-methoxypyridine
1-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-butyl-N-[2-(pyrazin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-({3-[methyl(quinolin-5-ylmethyl)carbamoyl]phenyl}amino)acetic acid
N-methyl-3-phenyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
(2H-1,3-benzodioxol-5-ylmethyl)({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)methylamine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]benzamide
2-[(E)-2-phenylethenyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-cyclopropyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-N-(pyridin-2-ylmethyl)acetamide
(3aS,7aR)-5-methyl-2-[(phenylcarbamoyl)carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
ethyl 2-[1-(2-oxo-6-phenyl-1,2-dihydropyridine-3-carbonyl)piperidin-2-yl]acetate
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1,3-oxazole-4-carboxamide
6-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
4-(4-fluorophenyl)-2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}-5-methylpyrimidine
1-[4-(piperidine-1-carbonyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
2-({[(3R,4R)-1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(1R,6S)-9-methyl-3-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
8-(1-benzofuran-2-ylmethyl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-(thiophen-2-ylmethyl)acetamide
1-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(1H-indazol-5-yl)urea
(3R,4S)-1-[(5,7-dimethyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]-4-propylpyrrolidin-3-amine
3-{4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}-1,2-dihydropyridin-2-one
4-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-imidazole-2-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-tert-butyl-N-(2-hydroxy-3-methoxypropyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl N-{1-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamoyl]ethyl}carbamate
N-(3-hydroxy-3-phenylpropyl)-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
2-(pyridin-4-ylmethyl)-9-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[4-(2-methylphenyl)-1,4-diazepan-1-yl]pyrimidin-4-amine
(2S)-3-(1H-imidazol-4-yl)-2-[(3-propyl-1H-pyrazol-5-yl)formamido]propanamide
3-(2-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-cyclopentyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one