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N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-4-sulfamoylbenzamide
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]pyridine-4-carboxamide
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
2-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-5-methylpyrazine
(2-methoxy-5-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenyl)methanol
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]furan-3-carboxamide
(2S,4R)-N-ethyl-4-[3-(ethylsulfanyl)propanamido]-1-(furan-2-carbonyl)pyrrolidine-2-carboxamide
1-(1H-imidazol-4-ylmethyl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
6-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
1-(2-methylpropyl)-6-(morpholin-4-yl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
2-amino-4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-6-propyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,4R)-4-phenyl-1-[2-(pyrrolidin-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
(3S,4R)-1-[1-(carbamoylmethyl)piperidine-4-carbonyl]-4-phenylpyrrolidine-3-carboxylic acid
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
(4aS,7aR)-1-[2-(2,6-dichlorophenyl)acetyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-({2-[1-(2-methoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(2,3-dihydro-1H-inden-2-yl)-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl][3-(5-methylfuran-2-yl)butyl]amine
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1'-[2-(pyridin-3-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
6-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyrazine-2-carboxamide
[(1-methyl-1H-pyrazol-4-yl)methyl]({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(propan-2-yl)amine
4-(1H-imidazol-1-ylmethyl)-2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazole
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidine-3-carbonitrile
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
4-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[(2,3,6-trifluorophenyl)methyl]butanamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(3,3,4,4-tetrafluorobutyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1H-indazole
2-methyl-6-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydropyridazin-3-one
3-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}propanamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-[benzyl(methyl)amino]-N-(2,3-dihydroxypropyl)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(2H-1,3-benzodioxol-5-yl)propanamide
ethyl 4-[1-(2-fluorophenyl)-3-(1-hydroxycyclopentyl)prop-2-yn-1-yl]piperazine-1-carboxylate
1-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one
3-methyl-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-1H-pyrazole-5-carboxamide
N-(4-fluorophenyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperazine-2-carboxamide
1-({3-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
1-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(2,3-dimethylphenoxy)ethan-1-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(3,3,4,4-tetrafluorobutyl)-3,6-diazabicyclo[3.2.2]nonane
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
1-(carbamoylmethyl)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]piperidine-3-carboxamide
5-chloro-6-[5-chloro-2-(propan-2-yloxy)phenyl]-2-methylpyrimidin-4-ol
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-(cyclohex-1-en-1-ylmethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 4-(2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetyl)piperazine-1-carboxylate
6-(4-fluorophenyl)-N-(3-methylbutyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid