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3-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}benzoic acid
1-(cyclopropylmethyl)-4-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(propan-2-yl)-1,4-diazepane
1-{2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-2-{4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}-4-(thiophen-2-ylmethyl)piperazin-2-one
3-{1-methyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
2-{4-[2-(ethylamino)pyrimidine-5-carbonyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-(pyrrolidin-1-yl)butanamide
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
ethyl 2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
4-({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)pyridine
2-chloro-3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
8-{5-[5-(methoxymethyl)furan-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}quinoline
(3aS,6aS)-2-(oxan-4-yl)-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N'-(3-ethylphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]butanediamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1,2-oxazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]acetamide
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-1H-indazole-3-carboxamide
N-(2-acetylphenyl)-3-{[2-(pyridin-2-yl)ethyl]amino}propanamide
3-(3-methoxyphenyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-4-carboxamide
2-(3-chloro-2-fluorophenyl)pyridine-3-carbonitrile
4-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-1-phenylbutan-1-one
N-[2-(diethylamino)ethyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
(2R)-N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)oxolane-2-carboxamide
(3S,4S)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-(2-methanesulfonylethyl)-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazine
1-(furan-2-ylmethyl)-3-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}piperidine
2-[1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]-1,3-benzothiazole
1-({5-[(2,4-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(2-methyl-4-{[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
2-[1-(2-methylpropyl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
1-methyl-3-(propan-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1H-pyrazole-5-carboxamide
(3R,5S)-N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(3-methoxypropanoyl)piperidin-3-yl]propanamide
3-methoxy-1-{2-[2-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
[3-(3-methylbut-2-en-1-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]methanol
7-(4-methoxy-2-methylbenzoyl)-2-methyl-2,7-diazaspiro[4.5]decane
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1,4-diazepane
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(2-methylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-methylfuran-2-yl)methyl]-3-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]propanamide
4-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperidin-3-yl)pyrimidine
(2S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-cycloheptyl-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1-oxaspiro[4.5]decan-2-one
{[3-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide