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ethyl 4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperazine-1-carboxylate
6-[(4-chlorophenyl)amino]-1-[2-(ethylsulfanyl)ethyl]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
3-{1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
6-cyclopropyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidin-4-amine
2-methyl-6-(2-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
N-[3-(4-methoxyphenyl)propyl]-6-(1H-pyrazol-4-yl)pyridine-3-carboxamide
1-[3-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-2-yl)ethane-1,2-dione
3-{[2-(ethylamino)pyrimidin-5-yl]formamido}-3-(4-fluorophenyl)propanoic acid
4-(5-fluoro-2-methylphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3R)-1-(5-fluoro-4-methoxypyrimidin-2-yl)-3,4,4-trimethylpyrrolidin-3-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(3R,4S)-4-({[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}(ethyl)amino)oxolan-3-ol
4-chloro-1-methyl-3-{1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-indazole
1-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-ethyl-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-(3,4-dimethylphenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-amine
N-methyl-2-{5-methyl-3-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}acetamide
(4aS,7aR)-1-(2-hydroxy-3-methoxybenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{2-[4-(morpholin-4-yl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-(1-benzylpiperidin-4-yl)-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
1-[4-(1-methylpiperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2,2-diphenylethan-1-ol
2-methyl-4-{3-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecane-3-carbonyl]phenyl}butan-2-ol
2-(4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}morpholin-3-yl)acetamide
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N4-[(3S)-1-benzylpyrrolidin-3-yl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(2-methoxyphenoxy)propyl]-N-methylacetamide
3-chloro-4-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
(4aS,7aR)-1-[(8-chloroquinolin-2-yl)methyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(5-amino-1H-pyrazole-3-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
7-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-(cycloheptylamino)-N-methylpyrrolidine-2-carboxamide
methyl[(1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]amine
9-[5-(methoxymethyl)furan-2-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(4aS,8aR)-6-(2-methyl-1H-pyrrole-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-2-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
2-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(3S,4R)-3-benzyl-4-methyl-1-(pyrimidin-2-yl)piperidin-4-ol
3-methyl-1-{4-[(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)sulfamoyl]phenyl}urea
2-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-methyl-N-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-(2-chlorophenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]furan-2-carboxamide
1-(butan-2-yl)-5-(pentan-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N-cyclopropylpiperazine-2-carboxamide
(2S,4S)-4-amino-1-(2,6-dimethoxypyrimidine-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
8-(3-methyl-1H-pyrazole-5-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
9-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide