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N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}pent-4-enamide
methyl 1-[3-(4-methoxyphenyl)-3-phenylpropanoyl]piperidine-4-carboxylate
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
15-methyl-12-(piperidine-1-carbonyl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
N-benzyl{[5-chloro-2-(1H-pyrazol-5-yl)phenyl]amino}sulfonamide
(3S,7S,8aS)-7-{[(2,5-difluorophenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-sulfonyl]-N-[2-(ethylsulfanyl)ethyl]benzamide
2-benzyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1,3-thiazole-4-carboxamide
(2S,4S)-4-cyclopentaneamido-N-ethyl-1-[(2-ethylphenyl)methyl]pyrrolidine-2-carboxamide
7-fluoro-N,2-dimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]quinoline-4-carboxamide
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})[(5-propyl-1H-pyrazol-3-yl)methyl]amine
1-{4-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
N-(2,3-dihydroxypropyl)-4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
N,3-diethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1H-indole-2-carboxamide
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
7-[3-(1H-pyrazol-4-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
6-chloro-3-fluoro-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}imidazo[1,2-a]pyridine
N,N-dimethyl-2-(2-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}phenoxy)acetamide
3-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}phenol
1-(2-hydroxyethyl)-1-[(5-methylthiophen-2-yl)methyl]-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
6-[1-(7-fluoro-2-methylquinoline-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
(3aS,6aR)-5-cyclopentyl-3-[(3,4-dimethoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(3-fluorophenyl)methyl]-4-(3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazin-2-one
2-({[(3R,4R)-1-(2,3-difluoro-6-methoxybenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[(4-acetylmorpholin-2-yl)methyl]-1-[4-chloro-2-(trifluoromethyl)phenyl]urea
2-(phenoxymethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
(2R,4S)-4-hydroxy-1-[(2E,6Z)-nona-2,6-dien-1-yl]piperidine-2-carboxylic acid
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]acetamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(2-fluoro-4,5-dimethoxyphenyl)pyridine-3-carbonitrile
(4S)-3-[(4-methoxypyridin-2-yl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
11-[2-(prop-2-en-1-yloxy)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
8-(3-methylfuran-2-carbonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
2-[3-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenoxy]acetamide
1-(2-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-ethyl-N-[2-(4-fluorophenyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
3-chloro-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}phthalazine
4-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(1,4-dimethylpiperazin-2-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
1-cyclopentyl-4-[(4-fluoro-3-methoxyphenyl)methyl]piperazin-2-one
6,6-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-5-oxothiomorpholine-3-carboxamide
2-cyclohexyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-(4-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}thiophen-2-yl)ethan-1-one