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N-[2-(furan-2-yl)ethyl]-3-[(1H-imidazol-2-ylmethyl)sulfamoyl]benzamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-methyl-4-(3-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)butan-2-ol
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-[(3,4-dimethylphenyl)methyl]-4-(2-methylpyridin-4-yl)piperazin-2-one
3-(6-methoxynaphthalene-2-carbonyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
3-[5-(2-amino-6-methylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
2-[3-(pyridin-4-yl)-5-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl]acetic acid
6-[4-(3-cyanopyridin-2-yl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-3-carboxylic acid
2-amino-6-(indolizin-2-yl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
4-[6-(trifluoromethyl)pyridin-2-yl]benzonitrile
1-(3-fluorobenzenesulfonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
5-{[3-cyclopentyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-N-butyl-1-cyclopropyl-6-oxopiperidine-3-carboxamide
2-{[(3R,4S)-3-cyclobutaneamido-4-propylpyrrolidin-1-yl]methyl}benzoic acid
N-(4-ethoxyphenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-benzyl-5-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyrimidin-2-amine
N-[1-(pentan-2-yl)-1H-pyrazol-5-yl]-4-(pyridin-3-yl)piperazine-1-carboxamide
N2-[(2-methoxyphenyl)methyl]-N2-(prop-2-en-1-yl)pyrrolidine-1,2-dicarboxamide
9-(2,6-dimethylpyrimidine-4-carbonyl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aS)-2-[(1-methyl-1H-imidazol-5-yl)methyl]-decahydroisoquinolin-4a-ol
2-(4-cyclopropanecarbonyl-3-fluorophenyl)benzamide
6-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-N-(propan-2-yl)pyrimidin-4-amine
2-(4-fluorophenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
4-methoxy-3-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}benzene-1-sulfonamide
1-{4-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-[2-(1H-indol-3-yl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-[(3-fluoro-4-methoxyphenyl)methyl]-2-methyl-1,4-oxazepane
1-(2-methoxyphenyl)-4-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]piperazine
2-{2-[({[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}carbamoyl)amino]phenyl}-N,N-dimethylacetamide
8-[(5-chlorothiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-[(3-ethoxy-4-hydroxyphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
(1-{5-[4-(hydroxymethyl)phenyl]-4-(4-methylphenyl)pyrimidin-2-yl}piperidin-4-yl)methanol
N-[(3-chloro-2-methylphenyl)methyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]cyclohexanamine
1-{3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]pyridin-2-yl}piperidin-3-ol
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
(1R,5S,8R)-3-(4-chloro-2-hydroxybenzoyl)-3-azabicyclo[3.2.1]octan-8-ol
1-cyclopropyl-N-[2-(3-methylthiophen-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-(6-methoxypyridin-3-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-methoxyphenol
3-{2-oxo-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
(2S,4S)-4-amino-1-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide