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N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
5-[1-(2-tert-butyl-1H-imidazol-1-yl)ethyl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
N-benzyl-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-ethyl-N-(2-methoxyethyl)-3-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-{2-[(4-ethoxypyrimidin-2-yl)amino]ethyl}-1,3-oxazinan-2-one
8-(1,3-benzothiazol-2-yl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
N-(butan-2-yl)-N-cycloheptyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-methylphenol
4-(2-hydroxy-6-methylquinolin-3-yl)-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(cyclopropylmethyl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-hydroxy-N-methyl-4-(methylsulfanyl)butanamide
N-methyl-N-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[(3R,5R)-5-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine-3-carbonyl]morpholine
4-(1,2,4-oxadiazol-3-yl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine
1-[2-(4-methoxyphenyl)ethyl]-5-(6-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-N-methylpyrrolidine-3-carboxamide
(3aS,6aS)-5-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
6-(3-fluoro-4-methoxyphenyl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
2-methoxy-5-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]pyrimidine
7-(oxan-4-yl)-2-[2-(pyridin-2-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}piperidin-2-one
(2S)-N-[(3-phenylphenyl)methyl]-1-(piperidin-4-yl)pyrrolidine-2-carboxamide
4-(1H-imidazol-1-yl)-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-6-(piperidin-3-yl)pyrimidin-4-amine
1-(3-chloro-5-methoxybenzoyl)-3-(2-methoxyphenoxy)azetidine
(2R,3R,6R)-5-(2-ethoxypyridine-3-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-4-[1-(4-cyanophenyl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
(3aS,6aR)-5-(3-methylbenzoyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 2-{4-[(2-fluorophenyl)methyl]-5-oxo-1,4-diazepane-1-carbonyl}benzoate
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
methyl 8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-ethoxyphenyl)-3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]urea
1-(4-methoxyphenyl)-5-methyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(methylamino)ethyl]piperidine-3-carboxamide
3-{1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}phenol
{[1-(morpholin-4-yl)cycloheptyl]methyl}[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-(4-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
methyl 2-(cyclopropylsulfamoyl)-6-[3-(trifluoromethyl)benzoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-chloro-2-{[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]methyl}phenoxy)acetamide
4-{5-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
1-methyl-4-(quinoxalin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1,7-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
7,8-dimethyl-3-(2,2,6,6-tetramethylpiperidin-4-yl)-3,4-dihydroquinazolin-4-one
2-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-7-ethyl-2,7-diazaspiro[4.5]decan-6-one