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(1S,5R)-3-[(5-acetylthiophen-3-yl)methyl]-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
(2S,4S)-4-amino-1-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
3-(1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
2-(morpholin-4-yl)-1-(1,4-oxazepan-4-yl)-2-(pyridin-3-yl)ethan-1-one
N-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}acetamide
4-[4-(4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]morpholine
N-[2-(1H-imidazol-4-yl)ethyl]-4-(pyrrolidin-1-ylmethyl)benzamide
2-[2-(1-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
(1S,5R)-6-benzyl-3-(3,3,3-trifluoropropanoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(pyridin-4-yl)-7-[2-(pyrrolidin-1-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-3-[2-(methylamino)pyridine-4-carbonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-benzylpiperidin-4-yl)-5-(3-chlorophenyl)-1,2,4-triazin-3-amine
2-{9-[2-(3-hydroxyphenyl)acetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
2-(4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[(3-methoxyphenyl)methyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}propanamide
N-cyclopropyl-3-{1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]piperidin-4-yl}propanamide
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-carbonyl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-benzyl-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,5-dimethyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
2-hydroxy-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyridine-3-carboxamide
4-[4-(piperidine-1-carbonyl)phenoxy]-1-(pyrrolidine-1-carbonyl)piperidine
3-[5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-hydroxy-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzoic acid
(3S)-4-(3-chlorothiophene-2-carbonyl)-3-ethylmorpholine
2-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazine
4-benzyl-3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-(1,3-thiazol-2-ylmethyl)piperidin-4-amine
2-(1H-indol-5-yl)-5-methoxybenzoic acid
2-(3-chloro-4-hydroxyphenyl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}ethan-1-one
5-[1-(3-methylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-[3-(4H-1,2,4-triazol-4-yl)phenyl]quinoline
(1S,4S)-2-(4-chloro-2-methoxy-5-methylphenyl)-5-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(4,5-dimethylfuran-2-yl)-1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazole
{[3-(cyclopentyloxy)phenyl]methyl}(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
1-cyclohexyl-N3-methyl-4-oxo-N5-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-(4-chlorophenyl)-1-[3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-4-ol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(3-hydroxyazetidin-1-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
2-{[2-amino-6-(2-ethoxyphenyl)pyrimidin-4-yl]amino}ethan-1-ol
3-{5-[3-(methylsulfanyl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-yloxy)propan-1-one
1,3-dimethyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-methyl-2-oxo-8-[2-(trifluoromethyl)benzoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-hydroxy-3-{[4-methoxy-4-(prop-2-en-1-yl)piperidin-1-yl]methyl}-1-(2-phenylethyl)piperidin-2-one
1-cyclopropyl-4-{[(5-ethylpyrimidin-2-yl)amino]methyl}pyrrolidin-2-one
(2S)-2-hydroxy-1-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one