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5-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(2-methoxyphenyl)ethyl]-4-phenyl-1H-imidazole
1-(difluoromethyl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
[1-(2-chloro-5-fluorobenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
1-(4-methoxyphenyl)-4-(1-propylpiperidin-4-yl)piperazine
1-ethyl-4-[1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N,6-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-(azocan-1-yl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
(3aS,6aS)-2-{[2-(ethylamino)pyrimidin-5-yl]methyl}-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carboxylic acid
1,4,6-trimethyl-2-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-{1-oxa-7-azaspiro[3.5]nonane-7-sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(trifluoromethyl)benzamide
1-[(2-methoxyphenyl)methyl]-5-(4-methoxypiperidine-1-carbonyl)piperidin-2-one
3-[(3R,4S)-1-[2-(3-chlorophenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-{[3-({1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-4-yl}oxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
3-(dimethylamino)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}benzamide
1-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-methylpyrazin-2-yl)methyl]acetamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]quinoxaline-6-carboxamide
5-[(dimethylamino)methyl]-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)furan-2-carboxamide
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrimidin-2-amine
N-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)acetamide
1-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)ethan-1-ol
3-{3,5-dimethyl-4-[2-(2-methylpropoxy)phenyl]-1H-pyrazol-1-yl}propanamide
2-(morpholin-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-ethyl-1,3,4-oxadiazol-2-amine
1-methyl-5-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrrole-2-carboxamide
5-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-[(4-fluorophenyl)methyl]-3-(2-methoxyacetamido)-N-(prop-2-en-1-yl)benzamide
1-(2,6-dimethylpyridin-4-yl)-4-[2-(methylsulfanyl)benzoyl]piperazine
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2-methoxyphenyl)methyl]piperidine
2-[5-(2,6-dichlorophenoxymethyl)-1,2,4-oxadiazol-3-yl]pyrazine
2-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxo-N-(propan-2-yl)acetamide
2-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-3-carbonitrile
[(3R,4R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[3-(pyrrolidin-1-yl)propyl]acetamide
4-hydroxy-4-(hydroxymethyl)-N-[2-(3-methylphenoxy)phenyl]azepane-1-carboxamide
4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
1-ethyl-4-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]piperazine
(1R,5S,6S)-6-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
2-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-4-methoxyphenol
(1R,2S)-N1-butyl-N2-(1H-1,2,3,4-tetrazol-5-ylmethyl)cyclohexane-1,2-dicarboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
ethyl 2-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-2-yl)acetate
3-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one