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2,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylquinoline-3-carboxamide
N-methyl-1-(3-phenylpropyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N4-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-[4-(cyclopentylmethyl)piperazine-1-carbonyl]isoquinoline
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
6-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
5-(methanesulfonylmethyl)-1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
(1S,5R)-3-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl({[5-(morpholine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})(1,2-oxazol-3-ylmethyl)amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
1-ethyl-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
1-methyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-3-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}urea
4-[4-(4-benzylpiperazine-1-carbonyl)piperidin-1-yl]-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(dimethylamino)ethyl]-2-(1H-imidazol-1-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
N-cyclopropyl-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
6-(1-methyl-1H-imidazol-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyridazin-3-amine
{3-[(3,5-dimethyl-1H-indol-2-yl)methyl]-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)benzoic acid
N-(1,3-benzoxazol-2-ylmethyl)-5-(2,6-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-(2,5-dimethoxyphenyl)-1-(oxan-4-yl)pyrrolidine
(4S)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)ethan-1-one
N-[3-(4-fluorophenyl)phenyl]-1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidine-3-carboxamide
N-ethyl-6-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl}pyridine-3-carboxamide
N-[(2,4-dihydroxyphenyl)methyl]-1-(2-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
5-[2-(benzyloxy)phenyl]pyrimidin-2-amine
1-[1'-(dimethyl-1,3-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
5-methoxy-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrimidin-2-amine
1-{2-[1-(4-methylphenyl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
2,5,6-trimethyl-N-[1-(6-methylpyridin-3-yl)ethyl]pyrimidin-4-amine
[(3R,4R)-1-(2,6-dimethoxypyridine-3-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(3-methyl-1H-pyrazol-1-yl)-1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-(2,5-dimethoxyphenyl)-N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-N-methylbenzene-1-sulfonamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxy-1-oxopropan-2-yl}acetamide
(3R,4S)-1-[(3-chloro-4,5-dimethoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-cyclopropyl-1-(4-methanesulfonylphenyl)-5-(2-methoxy-5-methylphenyl)-1H-1,2,4-triazole
methyl 2-[3-(4-methoxyphenyl)-3-phenylpropanamido]acetate
propyl 2-(5-methoxy-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-(3-propoxypiperidin-1-yl)propan-1-one
1-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-N-methylpyrrolidine-3-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
N4,6-dimethyl-N2-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyrimidine-2,4-diamine