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(4-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1-methylpiperazin-2-yl)methanol
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
(1S,5R)-6-[(2-methoxynaphthalen-1-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
4-chloro-N,1-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
2-{[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl](thiophen-2-ylmethyl)amino}ethan-1-ol
(2S,3R)-2-({5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)-3-hydroxybutanamide
3,3,3-trifluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)propanamide
1-(oxolane-2-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4,4,4-trifluorobutan-1-one
3-(6-methoxynaphthalene-2-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
N-[2-(oxan-3-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-phenyl-1H-pyrazole
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(naphthalen-2-yl)piperazine
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-1H-1,2,4-triazole-5-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-{[1-(3-fluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}cyclopropanamine
N-(1-methoxypropan-2-yl)-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
ethyl 1-{[4-(4-acetyl-1,4-diazepan-1-yl)quinazolin-2-yl]methyl}piperidine-3-carboxylate
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenoxybutan-1-one
2-({[4-(methylsulfanyl)phenyl]methyl}({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl})amino)ethan-1-ol
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](2-methoxyethyl)amine
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
4-methyl-7-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)-2H-chromen-2-one
ethyl 4-[3-(benzylcarbamoyl)phenoxy]piperidine-1-carboxylate
N-ethyl-N-(2-hydroxyethyl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(4aS,8aR)-6-(3-fluoropyridin-2-yl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
4-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
(3S,4R)-4-(3-fluorophenyl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidine-3-carboxylic acid
(2S,4R)-1-(1-ethylpiperidin-4-yl)-N-methyl-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
1-(4-fluorophenyl)-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-1,4-diazepane
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(methylamino)pyridine-4-carboxamide
ethyl 1-(2-methoxypyridine-3-carbonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(1R,4S)-N-ethyl-1,7,7-trimethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
1-[2-methoxy-4-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
[(5-fluoro-1-methyl-1H-indol-2-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
2-(but-3-en-1-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-{3-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}morpholine
4-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]pyrimidine
3-[(dimethylamino)methyl]-1-[3-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-ol
6-(1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidin-3-yl)pyrimidin-4-ol
(3S)-N,N-dimethyl-1-(9H-purin-6-yl)azepan-3-amine
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-methylbenzoyl)piperidin-3-yl]propanamide
3-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}propanoic acid
1-[2-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
5-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-2-(4-methylphenyl)pyrimidin-4-ol
(3S,4R)-4-(4-fluorophenyl)-1-[2-(morpholin-4-yl)ethyl]pyrrolidine-3-carboxylic acid
(2R,3R)-3-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol