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2-(2-fluoro-5-methoxyphenyl)-2-[methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-propoxypiperidine
2-[(5-methylpyrazin-2-yl)methyl]-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1H-imidazol-2-yl)phenol
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
(3aR,6aR)-2-[(5-ethylpyridin-2-yl)methyl]-5-(thiophen-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-phenyl-2-[2-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-(3-acetylphenyl)-3-[methyl(2-phenylethyl)amino]piperidine-1-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
7-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
4-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-methylpyridine
2-ethyl-4-methyl-5-[(3R,4R)-1-methyl-4-(pyrrolidine-1-carbonyl)pyrrolidin-3-yl]-1H-imidazole
2-ethyl-6-[2-(3-methylphenyl)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-[1-(hydroxymethyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-(2-ethoxyethyl)-1,7-dimethyl-1H-indole-2-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
1-(4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)-2-phenoxyethan-1-one
N-(5-methyl-4H-1,2,4-triazol-3-yl)-4-(4-phenylphenyl)piperazine-1-carboxamide
2-(4-{[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
1-(1-benzyl-1H-pyrazole-4-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
1-(2-{7-methyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
3-{[ethyl(4-hydroxybutyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
2-(2-hydroxyethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
3-ethyl-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
1-{4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
4-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-5,6,7,8-tetrahydroquinazolin-2-amine
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine
dimethyl(1-{3-[1-methyl-3-(pyridin-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}ethyl)amine
1-[2-(1-{2-[4-(hydroxymethyl)phenyl]acetyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
4-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]-2,1,3-benzothiadiazole
methyl 3-[(cyclobutylformamido)methyl]-5-(4-fluorobenzenesulfonamido)benzoate
1-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)pyrimidine-4-carboxamide
5-methyl-4-{[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
2-[(5-methylpyrazin-2-yl)methyl]-9-[3-(methylsulfanyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-{[5-(naphthalen-2-yl)-1,2,4-triazin-3-yl]amino}piperidine-1-carboxylate
1-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
1-(1,3-benzothiazol-2-yl)-N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
(4aR,8aR)-2-(5-ethylthiophene-3-carbonyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
1-(4-{5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperazin-1-yl)ethan-1-one
3-(6-methoxypyridin-3-yl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
7-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
1-[1-(5-phenyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]piperidin-4-ol
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-(1,2-oxazol-5-yl)thiophene-2-sulfonamide
1-[4-(ethylamino)pyrimidin-2-yl]-3-phenylpyrrolidin-3-ol
N-cyclopropyl-1-[1-(4-methylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
(3S,4S)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidine-3,4-diol