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2-(2-phenyl-1H-imidazol-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-(1H-pyrrole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-(2,4,5-trifluorophenyl)pyridine-3-carbonitrile
1-(2-{[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-3-ol
N-cyclopropyl-4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperazine-2-carboxamide
3-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]propyl acetate
2-(3-chloro-4-hydroxyphenyl)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
3-[5-(hydroxymethyl)furan-2-carbonyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(3R,4R)-1-(1-benzofuran-2-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
3-propyl-N-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-pyrazole-5-carboxamide
methyl (2S,4S)-4-{[(2,2-dimethylpropoxy)carbonyl]amino}-1-methylpyrrolidine-2-carboxylate
1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-3-propylpiperidine-3-carboxylic acid
8-[1-(4-methylphenyl)cyclopropanecarbonyl]-1-oxa-8-azaspiro[4.5]decane
3,5-dimethyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,2-oxazole-4-carboxamide
2-[6-hydroxy-4-(2-methanesulfonylethyl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]-3-methylpiperidine-3-carbonitrile
3-cyclopropyl-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
(3aR,5R,6S,7aS)-2-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-octahydro-1H-isoindole-5,6-diol
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2,2-diphenylacetamide
N,5-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(1-phenylcyclopropyl)-1,3-oxazole-4-carboxamide
4-(2,5-dimethoxyphenyl)-2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenol
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-[2-(dimethylamino)ethyl]piperidin-4-amine
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-ethylpyrimidine
3-{4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carbonyl}-1,2-dihydroquinoxalin-2-one
N4-{[1-(methoxymethyl)cyclopropyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
7-cyclohexyl-2-(5-hydroxypyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(6-methylquinolin-5-yl)methyl]acetamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-ol
4-({3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzoic acid
4-[(4-{[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)sulfonyl]morpholine
methyl 4-[(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)carbamoyl]piperazine-1-carboxylate
2-phenyl-N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
3-(3-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-hydroxyphenyl)propanamide
(1R,7S)-6-(4-ethyl-3-oxopiperazine-1-carbonyl)-3-[(3-methylphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-(2-chlorophenyl)-N,2-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}furan-3-carboxamide
1-[3-(4-fluorophenyl)benzoyl]azepan-4-amine
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(6-chloropyridazin-3-yl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
methyl 4-[(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carbonyl)amino]benzoate
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
2-(4-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
2-hydroxy-3-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
3-(1H-indol-3-yl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
N-{2-[(2-ethylpyrimidin-5-yl)formamido]ethyl}-2,2,2-trifluoroacetamide