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methyl 4-{[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}butanoate
3-[5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-(3,4-difluorophenyl)-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}propan-1-one
6-methyl-4-{3-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-fluoro-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-cyclohexyl-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)isoquinoline-5-carboxamide
4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}-N-propylpiperidine-1-carboxamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3,6-trifluorophenyl)methyl]piperidine
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3-(azepane-1-carbonyl)-1-ethyl-N-[(2-fluorophenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[1-(hydroxymethyl)cyclopentyl]amino}-N-(1-phenylethyl)propanamide
1-(4-methoxy-2,5-dimethylphenyl)-1H-1,3-benzodiazole
4-(4-fluoro-2-methylphenoxy)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
N-[2-(2-ethoxyethoxy)phenyl]-4,4-difluoropiperidine-1-carboxamide
{1-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]piperidin-3-yl}methanol
1-cyclopentyl-6-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide
5-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrimidin-2-amine
N-butyl-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-(carbamoylamino)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-9H-purine
1-(4-fluoro-3-methoxyphenyl)-3-[3-(propan-2-yloxy)propyl]urea
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
2,4-dimethyl-5-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrimidine
N,2,6-trimethyl-N-(thian-4-yl)quinoline-4-carboxamide
(3S,4S)-4-cyclopropyl-1-[4-(2,4-dioxoimidazolidin-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(4-methylpent-3-en-1-yl)piperidine
1-[(2S)-2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
1-[3-(methylsulfanyl)butyl]-4-(pyridin-3-yl)piperidin-4-ol
1-[1-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
8-(5-methyl-1,3-benzoxazol-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-{5-[(2S)-1-cyclohexanecarbonylpyrrolidin-2-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
ethyl 2-(1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}piperidin-2-yl)acetate
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3,5-dimethyl-1H-pyrrole-2-carboxamide
5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(methoxymethyl)pyrimidine
N-[2-(dimethylamino)ethyl]-2,3-difluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
1-(4-phenyl-1,3-thiazol-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(3-cyclopentylpropyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
(2R,3R,6R)-5-(3-fluorobenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(7-chloroquinolin-4-yl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(1H-indazol-1-yl)ethan-1-one
N-{2-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]quinolin-6-yl}acetamide
(3S,9aR)-3-(cyclohexylmethyl)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-cyclopentyl-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-4-carboxamide
4-[(4-cyclopentylpyrimidin-2-yl)amino]-1-propylpyrrolidin-2-one
(1S,5R)-6-propyl-3-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one