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1-(carbamoylmethyl)-N-cycloheptyl-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-(furan-3-ylmethyl)-5-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
3-chloro-N-(2-methoxyethyl)-4-({1-[1-(4-methylphenyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]-4-(methoxymethyl)piperidine
N-[2-(5-methylfuran-2-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({1-[(4-fluorophenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-2-methylbenzamide
2-({4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-8-fluoroquinoline-2-carboxamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
6-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-4-methyl-1H,2H,3H-pyrazolo[3,4-b]pyridin-3-one
1-(2-methyl-1,3-thiazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
5-(4-ethylbenzenesulfonyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(4aR,7aS)-6,6-dioxo-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-(1-{3-[(4-fluorophenyl)formamido]propanoyl}piperidin-3-yl)benzoic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
1-({4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-4-ol
N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(1R,2S,6R,7S)-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-4-azatricyclo[5.2.2.02,6]undecane
3-[(2-hydroxyethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]-1λ6-thiolane-1,1-dione
1-(2-methylphenyl)-4-[3-(pyridin-2-yl)propanoyl]piperazin-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-cyclopentyl-6-oxopiperidine-3-carboxamide
2-fluoro-6-methoxy-4-[(3-propylmorpholin-4-yl)methyl]phenol
N-ethyl-3-[1-(hydroxymethyl)-9-methyl-3,9-diazaspiro[5.5]undecan-3-yl]propanamide
2-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
3-(2-oxoimidazolidin-1-yl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
4-(2-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
3-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
ethyl 4-({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)piperidine-1-carboxylate
(3S,4R)-1-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(3-fluorophenyl)-4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1H-pyrazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-oxoazonan-1-yl)acetamide
7-methyl-4-(1,3-thiazol-4-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
(4aR,6R,8aS)-2-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
1-(2-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-methoxy-4-{[(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1H-pyrazole-3-carboxamide
2-[2-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-3-(2-oxopyrrolidin-1-yl)propanamide
2-(morpholin-4-ylmethyl)-N-[4-(trifluoromethoxy)phenyl]piperidine-1-carboxamide
4-(4-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-2-methylbutan-2-ol
N-(pyridin-2-ylmethyl)-3-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]oxy}benzamide
1-(1-benzylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
3-benzyl-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(1-ethyl-3-oxopiperazin-2-yl)acetamide
(3S,4R)-1-(1H-indazole-3-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
ethyl 1-[2-(furan-2-yl)-2-oxoacetyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-(benzyloxy)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][2-methyl-2-(piperidin-1-yl)propyl]amine