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(4aR,7aS)-1-[2-(2,2-dimethylmorpholin-4-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}piperazin-1-yl)propan-1-ol
5-(2-methoxyphenoxymethyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-3-carboxamide
1-{[({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)amino]methyl}cyclohexan-1-ol
(3R,5S)-5-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-3-ol
4-ethyl-3-{1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(1-methylpiperidin-2-yl)propanamide
5-[({[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(piperidin-1-yl)propan-1-one
3-(2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanamide
1-(oxolan-2-ylmethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
2-{1-[2-(oxolan-3-yl)ethyl]-1H-imidazol-2-yl}-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
1-(2-{1-cyclohexyl-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)pyrrolidin-2-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}acetamide
4-(2-methoxyphenoxy)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidine
N-(1-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
methyl 3-(2-cyclohexylacetamido)-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-(3-cyanophenyl)-3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}benzamide
2-methoxy-2-phenyl-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
N-(1H-indol-3-yl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
3-[(4-methyl-6-{[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amino}pyrimidin-2-yl)amino]phenol
methyl 4-{4-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperazin-1-yl}benzoate
2-(2-methyl-2-phenoxypropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2,4-difluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-[1-(3-phenylpropanoyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
8-(3-methoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-{[(2-fluoro-5-methoxyphenyl)methyl](methyl)amino}oxolan-3-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-(dimethylamino)-2-(4-methylphenyl)acetamide
8-(5-fluoropyrimidin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-amino-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}cyclopropane-1-carboxamide
N-{4-[3-(morpholin-4-ylmethyl)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
2-(azepan-1-yl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
2-(furan-2-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-oxoacetamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-(2-propylpyridine-4-carbonyl)pyrrolidine-2-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
4-{[4-(2-aminoethyl)phenyl]methyl}-5-methyl-1-(3-methylphenyl)piperazin-2-one
(5-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}furan-2-yl)methanol
2-amino-4-(furan-3-yl)-6-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
4-{[1-(1-ethyl-3-methylpiperidine-3-carbonyl)azetidin-3-yl]oxy}benzoic acid
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
1-[1'-(5-hydroxypyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-{1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(1S,3R)-3-amino-N-benzyl-N-(cyclobutylmethyl)cyclopentane-1-carboxamide
1-[3-oxo-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propyl]-1,2-dihydropyridin-2-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-(furan-2-ylmethyl)-N-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-amine
3-(pentan-2-yl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one