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3-methyl-2-propyl-4-[(1s,4s)-4-aminocyclohexyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 2-(morpholine-4-sulfonyl)-6-(naphthalen-2-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[2-(methylsulfanyl)ethyl]acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
(3S,5S)-1-benzyl-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-fluoro-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-5-sulfamoylbenzamide
8-chloro-5-methyl-1-(oxolan-3-yl)-[1,2,4]triazolo[4,3-a]quinoline
2-(2-ethylpyrimidin-5-yl)-7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
1-[4-(5-acetylthiophene-3-carbonyl)piperazin-1-yl]-2-phenoxyethan-1-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(methylamino)pyrimidine-5-carboxamide
(2E)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
7,7-dimethyl-2-[2-(pyridin-2-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,4S)-1-[3-(4-fluorophenyl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-chloro-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-(carbamoylmethyl)-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-3-carboxamide
1-cyclopentyl-3-(4-phenylpiperidine-1-carbonyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
2-(2-methoxyethoxy)-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
5-(3,3-diphenylpiperidine-1-carbonyl)-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-1,2-dihydropyridin-2-one
4-methoxy-6-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
1-(4-ethylpiperazin-1-yl)-3-{1-[1-(2-methoxyphenyl)propan-2-yl]piperidin-4-yl}propan-1-one
N-benzyl-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidine-4-carboxamide
1-ethyl-N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-3-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-(2-fluoroethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-N-cyclopropylpropanamide
4-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1,4-oxazepan-6-ol
N-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
methyl N-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}carbamate
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}prop-2-ene-1-sulfonamide
1-(3-hydroxypropyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
N-[(6-chloropyridin-3-yl)methyl]-5-ethyl-N,2-dimethylpyrimidin-4-amine
1-(2-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}pyrimidin-4-yl)pyrrolidin-3-ol
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-3,4-dimethoxybenzene-1-sulfonamide
1-(4-aminoazepan-1-yl)-2-(5-chloro-6-methyl-1-benzofuran-3-yl)ethan-1-one
N-methyl-6-oxo-4-[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(quinoline-3-carbonyl)piperidin-3-amine
5-(methoxymethyl)-N-(oxan-3-yl)thiophene-2-carboxamide
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
5-amino-N-[1-(4-fluorophenyl)piperidin-4-yl]-1H-pyrazole-3-carboxamide
5,6-dimethoxy-2-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydroisoquinolin-1-one
8-(furan-2-ylmethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)quinolin-8-ol
1-[(5-propylfuran-2-yl)methyl]-4-(pyridin-2-yl)piperazine
[(1S,3S,3aS,6aR)-3-[4-ethoxy-3-(hydroxymethyl)phenyl]-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
3-[8-(dimethyl-1,3-oxazole-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2-dihydropyrimidin-2-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide