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3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]propanamide
2-(2,5-dioxoimidazolidin-4-yl)-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
4-ethyl-3-({1-[(3-fluoro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-5-(propan-2-yl)-N-[3-(pyrrolidin-1-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(dimethylamino)ethyl]-N-[(2-methylphenyl)methyl]acetamide
1-[(4aR,8aR)-7-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-{4-[4-(piperidin-3-yl)benzoyl]piperazin-1-yl}-N-(propan-2-yl)acetamide
4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1-phenylpiperazin-2-one
2-ethyl-4-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-butyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2-(1,2-benzoxazol-3-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
1-[(3,4-dimethoxyphenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-[(2S,4R,6S)-2-(4-oxo-4H-chromen-3-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]amine
N-cyclopropyl-2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
2-(dimethylamino)-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
2-(1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1H-imidazol-2-yl)benzoic acid
2-{3-[3-(3-fluoro-4-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}-N-methylacetamide
2-[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]benzoic acid
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-4-yl}-2-phenylethan-1-ol
N-methyl-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
2-{[(3S,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
3-(3-phenylpropyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
3-{[2-(4,6-dimethylpyrimidin-2-yl)ethyl]sulfamoyl}-N,N-dimethylbenzamide
2-[(4aR,7aS)-4-(3-ethoxypropanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-({1-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperidin-4-yl}methyl)pyrrolidin-2-one
2-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
N-[(2-methoxynaphthalen-1-yl)methyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2R,3R)-3-amino-1'-(2-ethoxypyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aS,8aR)-6-(2-methylfuran-3-carbonyl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]acetamide
methyl 3-{4-[(1S,8R)-4-amino-5-cyano-3-azatricyclo[6.2.1.02,7]undeca-2,4,6-trien-6-yl]-1H-pyrazol-1-yl}propanoate
(2S,4S)-4-{4-[2-(2-cyclopentylacetamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}-N-methylpyrrolidine-2-carboxamide
6-methyl-5-[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]-2-(pyrimidin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-chloro-3-{[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]methyl}-1-methyl-1H-indazole
1-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-7-[2-(phenylsulfanyl)ethyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3R,4R)-1-cyclobutyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-3-yl)acetamide
N-[(3-methylphenyl)methyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
1-{3-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}isoquinoline
1-[(2-chloro-6-fluorophenyl)methyl]-3-cyclopropyl-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
1-methyl-2-{1-[(1-propylcyclobutyl)methyl]-1H-imidazol-2-yl}-1H-imidazole
2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
3-[4-hydroxy-4-(pyridin-3-yl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide