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methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(2-methoxyacetamido)methyl]benzoate
3-(3-methoxyphenoxy)-1-(3-methylbut-2-en-1-yl)azetidine
2-{[1-(3-phenylpropyl)piperidin-3-yl]amino}pyridine-3-carbonitrile
3-[(1-acetylpiperidin-4-yl)oxy]-N-(3-cyclopentylpropyl)-4-methoxy-N-methylbenzamide
2,6,8-trimethyl-N-(1-methyl-6-oxopiperidin-3-yl)quinoline-4-carboxamide
N-[1-(3-hydroxypropyl)-1H-1,3-benzodiazol-5-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[4-(3-methoxyphenyl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxamide
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N4-[(2,4-dimethoxyphenyl)methyl]-5-ethylpyrimidine-2,4-diamine
3-(2-oxo-2-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethyl)-4-[(4-phenylphenyl)methyl]piperazin-2-one
N-(2,4-difluorophenyl)-3-(2-phenylacetyl)piperidine-1-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3,5,7-trimethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
5-{[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-propylpyrimidin-2-amine
N-[(3,4-difluorophenyl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-[2-(1H-imidazol-4-yl)ethyl]pyrimidin-2-amine
3-(methoxymethyl)-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}piperidine
1-[(4-chlorophenyl)methyl]-4-(5-methoxyfuran-2-carbonyl)piperazine
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-(propan-2-yl)pyrimidin-4-amine
1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4S)-4-(4-{[(2,4-dichlorophenyl)formamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-3-yl}propanamide
N-{2-[5-methyl-4-({[4-(propan-2-yloxy)phenyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}pyridine-3-carboxamide
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
N-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)methanesulfonamide
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
(2S,4S)-4-amino-1-(2,2-diphenylacetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)piperazine
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-4-propylpyrimidine
N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-[4-(6-methoxypyrimidin-4-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
5-(2H-1,3-benzodioxole-5-carbonyl)-1-(cyclopropylmethyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-methylphenyl)-4-(quinoline-8-carbonyl)piperazin-2-one
N-(oxan-4-yl)-2-propyl-1,3-thiazole-4-carboxamide
3-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-{[(3-methylthiophen-2-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
1-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-ethylurea
N-[(1-cyclopentylpyrrolidin-3-yl)methyl]pyrimidin-4-amine
5-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-{1-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1H-1,2,3-triazol-4-yl}phenol
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydroquinoxalin-2-one
1-({1-[6-(6-methoxypyridin-3-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-[1-(pyridazine-3-carbonyl)piperidin-3-yl]benzoic acid
3-{[1-(3-fluorophenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
N-[(8-methoxyquinolin-5-yl)methyl]-N,5-dimethyl-1,3,4-oxadiazol-2-amine
N2-({4-[(dimethylamino)methyl]phenyl}methyl)-N2,N4-dimethylpyrimidine-2,4-diamine
4-[(3,4-difluorophenyl)methyl]-3-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
N-[2-(N-methylmethanesulfonamido)ethyl]-4-(1H-pyrrol-1-yl)benzamide
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one